SCHEMBL23836992

SCHEMBL23836992

NC(=O)c1nc(N2CCC(F)C2)ccc1N

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AXL P30530 9/20 0.41
MAP2K3 P46734 2/20 0.39
ROCK2 O75116 1/20 0.39
BTK Q06187 1/20 0.39
P2RX7 Q99572 2/20 0.38
MAP4K4 O95819 3/20 0.38
PRKCQ Q04759 1/20 0.37
HRH4 Q9H3N8 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22013143 0.81 MAPT (0.42) ROCK2
SCHEMBL14938741 0.77 MAP4K4 (0.40) MAP4K4HRH4HRH3
SCHEMBL31390848 0.73 HRH3 (0.56) HRH3
SCHEMBL20119411 0.72 SMPD3 (0.43) ROCK2PRKCQ
SCHEMBL17119925 0.69 P2RX7 (0.44) P2RX7
SCHEMBL31378785 0.69 MAP2K3 (0.51) AXLMAP2K3
SCHEMBL17626721 0.69 HRH3 (0.71) BTKHRH4HRH3
SCHEMBL18691294 0.69 HRH3 (0.71) BTKHRH4HRH3
SCHEMBL18691295 0.69 HRH3 (0.71) BTKHRH4HRH3
SCHEMBL22013122 0.69 MAP4K4 (0.53) MAP4K4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3882247-A1 SIX-MEMBERED AND SIX-MEMBERED HETEROCYCLIC COMPOUND AND USES THEREOF SERVING AS PROTEIN RECEPTOR KINASE INHIBITOR Shanghai Ennovabio Pharmaceuticals Co., Ltd. (CN) 2021-09-22 EP disclosed