Oxalic Acid

Oxalic Acid

SCHEMBL238506

Cc1nc(SCCN2CCCC2)nn1-c1ccc(Cl)c(Cl)c1.O=C(O)C(=O)O

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 12/20 0.49
KCNH2 Q12809 3/20 0.45
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
POLB P06746 1/20 0.43
BLM P54132 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL235551 0.99 SIGMAR1 (0.48) SIGMAR1KCNH2KDM4EALDH1A1SMN1; SMN2
Oxalic Acid SCHEMBL235579 0.99 SIGMAR1 (0.48) SIGMAR1KCNH2KDM4EALDH1A1SMN1; SMN2
Oxalic Acid SCHEMBL238732 0.94 SIGMAR1 (0.49) SIGMAR1KCNH2KDM4EALDH1A1SMN1; SMN2
SCHEMBL238868 0.94 SIGMAR1 (0.54) SIGMAR1KCNH2ALDH1A1POLBHTT
SCHEMBL238794 0.93 SIGMAR1 (0.53) SIGMAR1KCNH2ALDH1A1POLBHTT
SCHEMBL238110 0.93 SIGMAR1 (0.53) SIGMAR1KCNH2ALDH1A1POLBHTT
Oxalic Acid SCHEMBL239622 0.92 SIGMAR1 (0.49) SIGMAR1KCNH2KDM4EALDH1A1SMN1; SMN2
Oxalic Acid SCHEMBL235011 0.91 SIGMAR1 (0.50) SIGMAR1KCNH2KDM4EALDH1A1SMN1; SMN2
Oxalic Acid SCHEMBL239746 0.91 SIGMAR1 (0.62) SIGMAR1KCNH2KDM4EALDH1A1HTT
Oxalic Acid SCHEMBL238328 0.90 SIGMAR1 (0.50) SIGMAR1KCNH2KDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097394-B1 1,2,4-TRIAZOLE DERIVATIVES AS SIGMA RECEPTOR INHIBITORS ESTEVE LABOR DR (ES) 2013-12-25 EP claimed
US-8349878-B2 1,2,4-triazole derivatives as sigma receptor inhibitors LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2013-01-08 US claimed
US-20120004211-A1 1,2,4-TRIAZOLE DERIVATIVES AS SIGMA RECEPTOR INHIBITORS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2012-01-05 US claimed
EP-2097394-B1 1,2,4-TRIAZOLE DERIVATIVES AS SIGMA RECEPTOR INHIBITORS ESTEVE LABOR DR (ES) 2013-12-25 EP disclosed
US-8039497-B2 1,2,4-triazole derivatives as sigma receptor inhibitors LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2011-10-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120004211-A1 1,2,4-TRIAZOLE DERIVATIVES AS SIGMA RECEPTOR INHIBITORS SIGMAR1, TMEM97, OPRK1 SIGMAR1 1/4885KCNH2 2052/4885KDM4E 4169/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.