SCHEMBL2385144

SCHEMBL2385144

c1ccc2nc3ccncc3cc2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.65
HPGD P15428 3/20 0.65
GLA P06280 2/20 0.65
MAPT P10636 2/20 0.65
ACHE P22303 1/20 0.65
PDGFRB P09619 1/20 0.48
PDGFRA P16234 1/20 0.48
HTR3A P46098 1/20 0.48
CYP2A6 P11509 1/20 0.46
NQO2 P16083 1/20 0.44
EGFR P00533 1/20 0.43
PIK3CD O00329 1/20 0.43
PIK3CA P42336 1/20 0.43
CYP1A2 P05177 3/20 0.42
KDM4E B2RXH2 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
LMNA P02545 2/20 0.42
GAA P10253 2/20 0.42
CYP3A4 P08684 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acridine SCHEMBL1041524 0.89 MAPT (0.62) ALDH1A1HPGDGLAMAPTACHE
SCHEMBL255425 0.89 CLK1 (0.48) ALDH1A1HPGDGLAMAPTACHE
SCHEMBL4113492 0.87 MAPT (0.65) ALDH1A1HPGDGLAMAPTACHE
SCHEMBL30520081 0.84 CLK1 (0.47) ALDH1A1HPGDGLAMAPTACHE
SCHEMBL9392287 0.84 ALDH1A1 (0.56) ALDH1A1HPGDGLAMAPTACHE
SCHEMBL9394403 0.84 ALDH1A1 (0.56) ALDH1A1HPGDGLAMAPTACHE
SCHEMBL20272949 0.82 CLK1 (0.53) ALDH1A1HPGDGLAMAPTACHE
Acridine SCHEMBL28260005 0.81 ALDH1A1 (0.79) ALDH1A1HPGDGLAMAPTACHE
Acridine SCHEMBL1772714 0.81 ALDH1A1 (1.00) ALDH1A1HPGDGLAMAPTACHE
Acridine SCHEMBL8339 0.81 ALDH1A1 (1.00) ALDH1A1HPGDGLAMAPTACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-121135709-A Benzo [ b ] [1,6] naphthyridine compound and preparation method and application thereof 河北科技大学 2025-12-16 CN disclosed
CN-121135709-A Benzo [ b ] [1,6] naphthyridine compound and preparation method and application thereof 河北科技大学 2025-12-16 CN disclosed
EP-3386508-B1 CPAP-TUBULIN MODULE UNIV KOELN (DE) 2025-04-16 EP disclosed
US-11851427-B2 Phosphodiesterase inhibitors and uses thereof THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2023-12-26 US disclosed
US-20210130349-A1 NOVEL PHOSPHODIESTERASE INHIBITORS AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2021-05-06 US disclosed
US-10899756-B2 Phosphodiesterase inhibitors and uses thereof THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2021-01-26 US disclosed
US-10875856-B2 CPAP-tubulin module UNIVERSITAET ZU KOELN (DE) 2020-12-29 US disclosed
US-10626113-B2 Phosphodiesterase inhibitors and uses thereof THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2020-04-21 US disclosed
EP-3022205-B1 NOVEL PHOSPHODIESTERASE INHIBITORS AND USES THEREOF UNIV COLUMBIA (US) 2020-02-05 EP disclosed
US-20180362527-A1 CPAP-TUBULIN MODULE UNIVERSITAET ZU KOELN (DE) 2018-12-20 US disclosed
US-7498331-B2 Arthropod repellent pharmacophore models, compounds identified as fitting the pharmacophore models, and methods of making and using thereof UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 2009-03-03 US disclosed
WO-2008130515-A1 ANTI-CANCER AGENTS, COMPOSITIONS AND METHODS OF TREATING CANCERS ACB, LLC (US) 2008-10-30 WO disclosed
EP-1392289-A2 CASPASE INHIBITORS AND USES THEREOF Vertex Pharmaceuticals Incorporated (US) 2004-03-03 EP disclosed
WO-2002094263-A2 CASPASE INHIBITORS AND USES THEREOF VERTEX PHARMACEUTICALS INCORPORATED (US) 2002-11-28 WO disclosed
EP-1142892-A1 PROCESSES FOR THE PREPARATION OF NOVEL NAPHTHYRIDINE DERIVATIVES Nippon Kayaku Kabushiki Kaisha (JP) 2001-10-10 EP disclosed
US-4816464-A ANTIINFLAMMATORY AGENTS, ENZYME TISSUE DESTRUCTION AMERICAN HOME PRODUCTS CORPORATION (US) 1989-03-28 US disclosed
US-4816464-A ANTIINFLAMMATORY AGENTS, ENZYME TISSUE DESTRUCTION AMERICAN HOME PRODUCTS CORPORATION (US) 1989-03-28 US disclosed
US-4808612-A ANTIINFLAMMATORY AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1989-02-28 US disclosed
US-4751305-A ANTIINFLAMMATORY AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1988-06-14 US disclosed
US-4748246-A INTERLEUKIN ANTAGONISTS, ANTIINFLAMMATORY AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1988-05-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11851427-B2 Phosphodiesterase inhibitors and uses thereof PDE5A, PDE2A, PDE3A ALDH1A1 1252/4885HPGD 377/4885GLA 448/4885
US-10875856-B2 CPAP-tubulin module TUBB1, TUBA1C, TUBB ALDH1A1 3356/4885HPGD 4769/4885GLA 1610/4885
US-10899756-B2 Phosphodiesterase inhibitors and uses thereof PDE5A, PDE2A, PDE3A ALDH1A1 1252/4885HPGD 377/4885GLA 448/4885
US-10626113-B2 Phosphodiesterase inhibitors and uses thereof PDE5A, PDE2A, PDE3A ALDH1A1 1252/4885HPGD 377/4885GLA 448/4885
US-20210130349-A1 NOVEL PHOSPHODIESTERASE INHIBITORS AND USES THEREOF PDE5A, PDE2A, PDE3A ALDH1A1 1375/4885HPGD 477/4885GLA 438/4885
US-20180362527-A1 CPAP-TUBULIN MODULE TUBB1, TUBA1C, TUBB ALDH1A1 3356/4885HPGD 4769/4885GLA 1610/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.