SCHEMBL23856080

SCHEMBL23856080

O=C(N[C@@H](CN1CCC(F)(F)CC1)C(=O)O)OCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 1/20 0.57
TGM2 P21980 1/20 0.54
ITGB3 P05106 7/20 0.50
ITGA2B P08514 7/20 0.50
OPRK1 P41145 3/20 0.49
CTSK P43235 2/20 0.47
IDO1 P14902 1/20 0.47
TDO2 P48775 1/20 0.47
CCR1 P32246 1/20 0.46
PPARG P37231 1/20 0.46
PPARA Q07869 1/20 0.46
DPP4 P27487 1/20 0.46
KCNH2 Q12809 1/20 0.46
DPP7 Q9UHL4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23856082 1.00 HRH1 (0.57) HRH1TGM2ITGB3ITGA2BOPRK1
SCHEMBL5967157 0.83 HRH1 (0.59) HRH1ITGB3ITGA2BOPRK1CTSK
SCHEMBL15689075 0.82 ITGB3 (0.63) HRH1ITGB3ITGA2BOPRK1CTSK
SCHEMBL19924796 0.81 HRH1 (0.62) HRH1ITGB3ITGA2BOPRK1CTSK
SCHEMBL19924794 0.81 HRH1 (0.62) HRH1ITGB3ITGA2BOPRK1CTSK
SCHEMBL23135998 0.81 DPP4 (0.49) TGM2OPRK1CTSKCCR1DPP4
SCHEMBL5651104 0.77 KYNU (0.53) HRH1OPRK1CTSK
SCHEMBL7520315 0.76 HRH1 (0.62) HRH1ITGB3ITGA2BOPRK1PPARG
SCHEMBL16435200 0.76 HRH1 (0.52) HRH1ITGB3ITGA2BOPRK1CTSK
SCHEMBL27033000 0.76 DPP4 (0.45) TGM2OPRK1DPP4KCNH2DPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021191827-A1 TRIPEPTIDES DERIVATIVES FOR TREATING SARS-COV-2 INFECTIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2021-09-30 WO disclosed