SCHEMBL23889154

SCHEMBL23889154

CC(=O)c1cnc2cc(OCC(F)F)ccn12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
BRD9 Q9H8M2 3/20 0.38
BAZ2B Q9UIF8 2/20 0.38
CSF1R P07333 8/20 0.38
KIT P10721 1/20 0.36
MGLL Q99685 2/20 0.36
ABHD6 Q9BV23 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
SMARCA2 P51531 1/20 0.35
SMARCA4 P51532 1/20 0.35
PIK3CA P42336 1/20 0.35
ACACB O00763 3/20 0.34
TRIM24 O15164 1/20 0.34
TAF1L Q8IZX4 1/20 0.34
BAZ2A Q9UIF9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17438012 0.88 CSF1R (0.36) NPC1RAB9ACSF1RKITMGLL
SCHEMBL20646977 0.88 NPC1 (0.37) NPC1RAB9ACSF1RKITMGLL
SCHEMBL17437845 0.85 KDM4E (0.47) NPC1RAB9ACSF1RKITKDM4E
SCHEMBL24247822 0.84 CSF1R (0.37) NPC1RAB9ACSF1RKITMGLL
SCHEMBL24976174 0.80 PRMT5 (0.39) CSF1RMGLLABHD6KDM4EALDH1A1
SCHEMBL24976173 0.77 PDE8A (0.32) MGLLABHD6
SCHEMBL24247757 0.76 CSF1R (0.51) CSF1RKITKDM4E
SCHEMBL30935784 0.73 GAA (0.47) NPC1RAB9ACSF1RKDM4EALDH1A1
SCHEMBL24247829 0.73 NPC1 (0.63) NPC1RAB9ABAZ2BKITMGLL
SCHEMBL9941591 0.73 KDM4E (0.43) NPC1RAB9ACSF1RKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3402790-B1 SPIROHEPTANE SALICYLAMIDES AND RELATED COMPOUNDS AS INHIBITORS OF ROCK BRISTOL MYERS SQUIBB CO (US) 2021-10-06 EP disclosed