SCHEMBL23897367

SCHEMBL23897367

CCOC(=O)c1ccc(-c2ccnc(Nc3ccc(C)cc3)n2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.57
THRB P10828 1/20 0.57
RAB9A P51151 1/20 0.57
KMT2A Q03164 1/20 0.57
CAMK2D Q13557 3/20 0.56
MAPK8 P45983 1/20 0.54
MAPK10 P53779 1/20 0.54
JAK2 O60674 2/20 0.53
JAK3 P52333 2/20 0.53
PDPK1 O15530 1/20 0.53
SLC2A1 P11166 1/20 0.51
MAPT P10636 1/20 0.51
IKBKB O14920 3/20 0.50
ABL1 P00519 2/20 0.49
PDGFRB P09619 2/20 0.49
BCR P11274 2/20 0.49
PDGFRA P16234 2/20 0.49
ALK Q9UM73 1/20 0.49
CHUK O15111 1/20 0.49
KDR P35968 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4071652 0.91 MAPK8 (0.67) MEN1THRBRAB9AKMT2ACAMK2D
SCHEMBL2861035 0.91 MEN1 (0.55) MEN1THRBRAB9AKMT2ACAMK2D
SCHEMBL3947629 0.86 ABL1 (0.62) MEN1THRBRAB9AKMT2AMAPK8
SCHEMBL2866252 0.85 IKBKB (0.53) MEN1THRBRAB9AKMT2ACAMK2D
SCHEMBL2856029 0.84 JAK2 (0.72) CAMK2DMAPK8MAPK10JAK2JAK3
SCHEMBL14021582 0.83 GAA (0.58) CAMK2DJAK2JAK3IKBKBCHUK
SCHEMBL13911421 0.83 MAPK8 (0.77) CAMK2DMAPK8MAPK10JAK2JAK3
SCHEMBL4354673 0.83 CDK2 (0.65) MAPK8JAK2IKBKBCHUK
SCHEMBL3946636 0.83 RAB9A (0.57) MEN1THRBRAB9AKMT2AJAK2
SCHEMBL3947916 0.83 RAB9A (0.56) MEN1THRBRAB9AKMT2AJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220388967-A1 Phenyl Amino Pyrimidine Compounds and Uses Thereof SIERRA ONCOLOGY, INC. (US) 2022-12-08 US disclosed
US-20210309615-A1 PHENYL AMINO PYRIMIDINE COMPOUNDS AND USES THEREOF GLAXOSMITHKLINE LLC 2021-10-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210309615-A1 PHENYL AMINO PYRIMIDINE COMPOUNDS AND USES THEREOF JAK2, JAK1, JAK3 MEN1 4037/4885THRB 2768/4885RAB9A 3849/4885
US-20220388967-A1 Phenyl Amino Pyrimidine Compounds and Uses Thereof JAK2, JAK1, JAK3 MEN1 4037/4885THRB 2768/4885RAB9A 3849/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.