SCHEMBL2389903

SCHEMBL2389903

COC(C)NC(=O)c1c(-c2ccccc2O)ccc2c1C(C)=CC(C)(C)N2

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 10/20 0.43
PGR P06401 8/20 0.42
TDP1 Q9NUW8 2/20 0.41
ALDH1A1 P00352 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
CYP3A4 P08684 1/20 0.41
HSD17B10 Q99714 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
AR P10275 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2390300 0.90 NR3C1 (0.50) NR3C1PGRTDP1ALDH1A1CYP3A4
SCHEMBL2389909 0.82 PGR (0.42) NR3C1PGRAR
SCHEMBL2393569 0.82 PGR (0.45) NR3C1PGRTDP1ALDH1A1L3MBTL1
SCHEMBL2395174 0.80 PGR (0.43) NR3C1PGRTDP1ALDH1A1L3MBTL1
SCHEMBL2397569 0.79 PGR (0.45) NR3C1PGRTDP1ALDH1A1CYP3A4
SCHEMBL2393170 0.78 NPC1 (0.44) NR3C1PGRALDH1A1LMNASMN1; SMN2
SCHEMBL2389906 0.76 PGR (0.44) NR3C1PGRAR
SCHEMBL2395912 0.76 KDM4E (0.46) PGRTDP1ALDH1A1L3MBTL1HSD17B10
SCHEMBL2395158 0.75 PGR (0.45) NR3C1PGRTDP1ALDH1A1L3MBTL1
SCHEMBL2393220 0.74 PGR (0.46) NR3C1PGRTDP1ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8017775-B2 1-2-dihydroquinoline derivative having glucocorticoid receptor binding activity SANTEN PHARMACEUTICAL CO., LTD. (JP) 2011-09-13 US disclosed
US-20090326009-A1 Novel 1-2-Dihydroquinoline Derivative Having Glucocorticoid Receptor Binding Activity Santen Pharmaceutical Co., (JP) 2009-12-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090326009-A1 Novel 1-2-Dihydroquinoline Derivative Having Glucocorticoid Receptor Binding Activity NR3C1, NR3C2, NR5A1 NR3C1 1/4885PGR 201/4885TDP1 3515/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.