SCHEMBL23901080

SCHEMBL23901080

CC(C)(C)OC(=O)c1nn(C(c2ccccc2)(c2ccccc2)c2ccccc2)c2ccc(Br)cc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 9/20 0.50
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
GSK3B P49841 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
GABRA1 P14867 5/20 0.37
GABRG2 P18507 5/20 0.37
GABRB3 P28472 5/20 0.37
GABRA5 P31644 5/20 0.37
GABRA3 P34903 4/20 0.37
GABRA2 P47869 4/20 0.37
GABRA6 Q16445 4/20 0.37
GABRB2 P47870 2/20 0.37
PLA2G2A P14555 1/20 0.35
GABRA4 P48169 2/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31391671 1.00 ELANE (0.50) ELANECCNB2CDK1CCNB1GSK3B
SCHEMBL15059772 0.86 ELANE (0.47) ELANECCNB2CDK1CCNB1GSK3B
SCHEMBL14785602 0.85 ELANE (0.66) ELANEALDH1A1LMNAF2PLAU
SCHEMBL4143502 0.84 ELANE (0.45) ELANEPLA2G2A
SCHEMBL31391678 0.82 GABRA1 (0.39) ELANEGABRA1GABRG2GABRB3GABRA5
SCHEMBL4298389 0.80 ELANE (0.58) ELANEGABRA1GABRG2GABRB3GABRA5
SCHEMBL23901079 0.79 NTRK1 (0.34) ELANEGABRA1GABRG2GABRB3GABRA5
SCHEMBL23901077 0.79 PRMT5 (0.41) ELANEMAPK1F2PLAUKLKB1
SCHEMBL4142114 0.78 EGFR (0.47) ELANE
SCHEMBL4300088 0.77 ELANE (0.55) ELANECCNB2CDK1CCNB1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021197467-A1 MULTI-TARGET ANTI-TUMOR COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海华汇拓医药科技有限公司 2021-10-07 WO disclosed