SCHEMBL23901077

SCHEMBL23901077

CC(C)(C)OC(=O)c1nn(C(c2ccccc2)(c2ccccc2)c2ccccc2)c2ccc(B3OC(C)(C)C(C)(C)O3)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 2/20 0.41
WDR77 Q9BQA1 2/20 0.41
BACE1 P56817 1/20 0.35
BACE2 Q9Y5Z0 1/20 0.35
ROCK1 Q13464 1/20 0.35
AAK1 Q2M2I8 2/20 0.35
DGAT1 O75907 1/20 0.34
USP30 Q70CQ3 1/20 0.34
LIPG Q9Y5X9 2/20 0.33
P4HB P07237 1/20 0.33
LPL P06858 1/20 0.33
HIF1A Q16665 1/20 0.33
F2 P00734 3/20 0.33
F11 P03951 2/20 0.33
PRSS1 P07477 1/20 0.33
PRSS2 P07478 1/20 0.33
PRSS3 P35030 1/20 0.33
MAPK1 P28482 1/20 0.33
ELANE P08246 2/20 0.32
PLAU P00749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23901080 0.79 ELANE (0.50) F2MAPK1ELANEPLAUKLKB1
SCHEMBL31391671 0.79 ELANE (0.50) F2MAPK1ELANEPLAUKLKB1
SCHEMBL31636018 0.78 LPL (0.40) PRMT5WDR77BACE1ROCK1DGAT1
SCHEMBL19665906 0.78 LIPG (0.37) PRMT5WDR77BACE1ROCK1LIPG
SCHEMBL26390707 0.77 LPL (0.38) PRMT5WDR77BACE1ROCK1LIPG
SCHEMBL31391678 0.75 GABRA1 (0.39) MAPK1ELANE
SCHEMBL30581655 0.75 USP30 (0.46) PRMT5WDR77USP30
SCHEMBL26390720 0.75 USP30 (0.46) PRMT5WDR77USP30
SCHEMBL24137829 0.75 PRMT5 (0.43) PRMT5WDR77BACE1BACE2ROCK1
SCHEMBL26390694 0.74 USP30 (0.43) PRMT5WDR77USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021197467-A1 MULTI-TARGET ANTI-TUMOR COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海华汇拓医药科技有限公司 2021-10-07 WO disclosed