SCHEMBL23901109

SCHEMBL23901109

CN(CCN1CCCC1)c1ccc(C(=O)Nc2n[nH]c3ccc(C(CF)c4cc(F)ccc4F)cc23)c(NC2CCOCC2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
INSR P06213 19/20 0.52
ALK Q9UM73 19/20 0.52
IGF1R P08069 14/20 0.52
AURKA O14965 2/20 0.48
AURKB Q96GD4 2/20 0.48
DAPK3 O43293 2/20 0.48
MAP4K4 O95819 2/20 0.48
RET P07949 2/20 0.48
GRK5 P34947 2/20 0.48
CLK2 P49760 2/20 0.48
CDK7 P50613 2/20 0.48
PRKCQ Q04759 2/20 0.48
MST1R Q04912 2/20 0.48
PRKAA1 Q13131 2/20 0.48
LRRK2 Q5S007 2/20 0.48
CAMK1D Q8IU85 2/20 0.48
HIPK2 Q9H2X6 2/20 0.48
CLK4 Q9HAZ1 2/20 0.48
TBK1 Q9UHD2 2/20 0.48
MAP4K5 Q9Y4K4 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23901345 0.85 ALK (0.71) INSRALKIGF1RAURKAAURKB
SCHEMBL23901334 0.84 INSR (0.73) INSRALKIGF1RAURKAAURKB
SCHEMBL31391720 0.84 INSR (0.66) INSRALKIGF1RAURKAAURKB
SCHEMBL31391723 0.84 INSR (0.73) INSRALKIGF1RAURKAAURKB
SCHEMBL28999405 0.84 INSR (0.66) INSRALKIGF1RAURKAAURKB
SCHEMBL23901394 0.83 INSR (0.70) INSRALKIGF1RAURKAAURKB
SCHEMBL23901169 0.83 INSR (0.76) INSRALKIGF1RAURKAAURKB
SCHEMBL23901261 0.82 INSR (0.61) INSRALKIGF1RAURKAAURKB
SCHEMBL31391722 0.82 INSR (0.61) INSRALKIGF1RAURKAAURKB
SCHEMBL23901186 0.82 INSR (0.63) INSRALKIGF1RAURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916771-A Multi-target antitumor compound and preparation method and application thereof 浙江华海药业股份有限公司 2023-04-04 CN claimed
CN-115916771-A Multi-target antitumor compound and preparation method and application thereof 浙江华海药业股份有限公司 2023-04-04 CN disclosed
WO-2021197467-A1 MULTI-TARGET ANTI-TUMOR COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海华汇拓医药科技有限公司 2021-10-07 WO disclosed