SCHEMBL23901345

SCHEMBL23901345

CN(CCN1CCCC1)c1ccc(C(=O)Nc2n[nH]c3ccc(Cc4cc(F)ccc4F)cc23)c(NC2CCOCC2)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 20/20 0.71
INSR P06213 19/20 0.71
IGF1R P08069 14/20 0.64
AURKA O14965 2/20 0.58
AURKB Q96GD4 2/20 0.58
PLK4 O00444 2/20 0.58
DAPK3 O43293 2/20 0.58
NTRK1 P04629 2/20 0.58
PRKCG P05129 2/20 0.58
ROS1 P08922 2/20 0.58
FER P16591 2/20 0.58
LTK P29376 2/20 0.58
FRK P42685 2/20 0.58
MST1R Q04912 2/20 0.58
PTK2 Q05397 2/20 0.58
TNK2 Q07912 2/20 0.58
NTRK3 Q16288 2/20 0.58
MAP4K5 Q9Y4K4 2/20 0.58
JAK2 O60674 1/20 0.58
MAP4K4 O95819 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23901325 0.93 ALK (0.70) ALKINSRIGF1RAURKAAURKB
SCHEMBL23901394 0.91 INSR (0.70) ALKINSRIGF1RAURKAAURKB
SCHEMBL23901169 0.91 INSR (0.76) ALKINSRIGF1RAURKAAURKB
SCHEMBL23901109 0.85 INSR (0.52) ALKINSRIGF1RAURKAAURKB
SCHEMBL23901242 0.84 INSR (0.70) ALKINSRIGF1RAURKAAURKB
SCHEMBL23901162 0.84 INSR (0.75) ALKINSRIGF1RAURKAAURKB
SCHEMBL23901348 0.84 INSR (0.67) ALKINSRIGF1RAURKAAURKB
SCHEMBL23901241 0.84 INSR (0.67) ALKINSRIGF1RAURKAAURKB
SCHEMBL23901347 0.84 INSR (0.67) ALKINSRIGF1RAURKAAURKB
SCHEMBL590085 0.83 ALK (0.55) ALKINSRIGF1RAURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916771-A Multi-target antitumor compound and preparation method and application thereof 浙江华海药业股份有限公司 2023-04-04 CN claimed
CN-115916771-A Multi-target antitumor compound and preparation method and application thereof 浙江华海药业股份有限公司 2023-04-04 CN disclosed
WO-2021197467-A1 MULTI-TARGET ANTI-TUMOR COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海华汇拓医药科技有限公司 2021-10-07 WO disclosed