SCHEMBL23905308

SCHEMBL23905308

C[C@]1(C(N)=O)COc2c1cc(C(CN)C(F)(F)F)nc2-c1ccc(F)cc1

nearest known ligand 0.31

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.31
KCNH2 Q12809 2/20 0.30
NR1I2 O75469 1/20 0.30
SCN9A Q15858 1/20 0.30
CYP3A4 P08684 1/20 0.30
CFTR P13569 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
MAPK1 P28482 1/20 0.30
HSD17B10 Q99714 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23905423 1.00 GRM2 (0.31) GRM2KCNH2NR1I2SCN9ACYP3A4
SCHEMBL23196145 0.88 CNR2 (0.32) KCNH2
SCHEMBL23905511 0.88 CFTR (0.31) CFTR
SCHEMBL23905937 0.88 GABRA5 (0.33) GRM2KCNH2CYP3A4CFTR
SCHEMBL23905800 0.87 PTGS1 (0.31)
SCHEMBL24363612 0.87 PTGS1 (0.31)
SCHEMBL23196033 0.85 GRM2 (0.37) GRM2SCN9ACFTR
SCHEMBL23195908 0.85 MAPK14 (0.36) KDM4EALDH1A1
SCHEMBL23904779 0.82 ADORA2A (0.31)
SCHEMBL23904889 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021198981-A1 ANTIVIRAL COMPOUNDS AND USES THEREOF Janssen Biopharma, Inc. (US) 2021-10-07 WO disclosed