SCHEMBL23911836

SCHEMBL23911836

C=C(C)C1(C(=O)N(C)c2ccc(F)cc2)CC1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 3/20 0.37
TSHR P16473 1/20 0.37
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
PIK3CA P42336 1/20 0.34
POLQ O75417 1/20 0.34
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
APP P05067 1/20 0.33
TRPA1 O75762 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
DRD2 P14416 1/20 0.32
GPBAR1 Q8TDU6 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL307214 0.84 AGTR2 (0.43) AGTR2GAAMAPTPKMPOLQ
SCHEMBL18256941 0.83 AGTR2 (0.38) AGTR2GAAMAPTPKMPIK3CA
SCHEMBL22265647 0.83 GAA (0.39) AGTR2GAAMAPTPKMPIK3CA
SCHEMBL18542859 0.80 NOTUM (0.37) AGTR2TSHRGAAMAPTPKM
SCHEMBL14873216 0.80 AGTR2 (0.36) AGTR2GAAMAPTPKMPOLQ
SCHEMBL14817541 0.77 CYP3A4 (0.35) AGTR2GAAMAPTPKMPOLQ
SCHEMBL13927587 0.77 KMT2A (0.40) AGTR2TSHRGAAALDH1A1POLB
SCHEMBL13620068 0.77 AGTR2 (0.37) AGTR2TSHRPOLQSMN1; SMN2ALDH1A1
SCHEMBL30937116 0.74 GAA (0.37) AGTR2GAAMAPTPKMPIK3CA
SCHEMBL22766292 0.74 ALDH1A1 (0.41) TSHRGAAMAPTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593090-B1 C-MET MODULATOR PHARMACEUTICAL COMPOSITIONS EXELIXIS INC (US) 2021-10-13 EP disclosed