SCHEMBL23912896

SCHEMBL23912896

N=C(/C=N\NCCc1ccc2c(n1)NCCC2)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 15/20 0.52
ITGAV P06756 15/20 0.52
CXCR4 P61073 5/20 0.51
ITGB6 P18564 8/20 0.45
ITGB5 P18084 7/20 0.45
ITGB8 P26012 6/20 0.45
ITGB1 P05556 1/20 0.44
ITGA2B P08514 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20156036 0.82 ITGB3 (0.53) ITGB3ITGAVCXCR4ITGB6ITGB5
SCHEMBL20156312 0.81 ITGAV (0.52) ITGB3ITGAVCXCR4ITGB6ITGB5
SCHEMBL20156053 0.79 ITGB3 (0.54) ITGB3ITGAVCXCR4ITGB6ITGB5
SCHEMBL20156247 0.77 ITGAV (0.52) ITGB3ITGAVCXCR4ITGB6ITGB5
SCHEMBL20156008 0.76 ITGAV (0.53) ITGB3ITGAVCXCR4ITGB6ITGB5
SCHEMBL20156245 0.75 ITGAV (0.54) ITGB3ITGAVCXCR4ITGB6ITGB5
SCHEMBL20156242 0.74 CXCR4 (0.52) ITGB3ITGAVCXCR4ITGB6ITGB5
SCHEMBL26032494 0.74 ITGAV (0.54) ITGB3ITGAVCXCR4ITGB6ITGB5
SCHEMBL20156358 0.73 CXCR4 (0.52) ITGB3ITGAVCXCR4ITGB6ITGB5
SCHEMBL760607 0.73 ITGB3 (0.69) ITGB3ITGAVITGB6ITGB5ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538527-B1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2021-10-13 EP disclosed