SCHEMBL20156036

SCHEMBL20156036

N=C(/C=C\NCCc1ccc2c(n1)NCCC2)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.53
ITGAV P06756 14/20 0.53
CXCR4 P61073 6/20 0.52
ITGB5 P18084 6/20 0.45
ITGB6 P18564 6/20 0.45
ITGB8 P26012 6/20 0.45
ITGA2B P08514 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20156358 0.89 CXCR4 (0.52) ITGB3ITGAVCXCR4ITGB5ITGB6
SCHEMBL23912896 0.82 ITGB3 (0.52) ITGB3ITGAVCXCR4ITGB5ITGB6
SCHEMBL20156053 0.82 ITGB3 (0.54) ITGB3ITGAVCXCR4ITGB5ITGB6
SCHEMBL24521988 0.81 ITGB3 (0.63) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20156008 0.81 ITGAV (0.53) ITGB3ITGAVCXCR4ITGB5ITGB6
SCHEMBL20156245 0.81 ITGAV (0.54) ITGB3ITGAVCXCR4ITGB5ITGB6
SCHEMBL20156247 0.80 ITGAV (0.52) ITGB3ITGAVCXCR4ITGB5ITGB6
SCHEMBL26032494 0.79 ITGAV (0.54) ITGB3ITGAVCXCR4ITGB5ITGB6
SCHEMBL20156242 0.79 CXCR4 (0.52) ITGB3ITGAVCXCR4ITGB5ITGB6
SCHEMBL20156094 0.76 ITGAV (0.49) ITGB3ITGAVCXCR4ITGB5ITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538527-B1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2021-10-13 EP disclosed
WO-2018089358-A1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed