SCHEMBL23917111

SCHEMBL23917111

COCc1ccc(N2CCN(C)CC2)cc1OC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 1/20 0.55
HTR6 P50406 3/20 0.49
AGXT P21549 1/20 0.44
HTR3A P46098 1/20 0.44
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
KDM4E B2RXH2 4/20 0.44
GAA P10253 3/20 0.43
MAPT P10636 2/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
RECQL P46063 1/20 0.43
PTK2B Q14289 1/20 0.43
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
BLM P54132 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21566486 0.86 SIRT6 (0.59) SIRT6HTR6HTR3ADRD2DRD3
SCHEMBL8325286 0.82 AGXT (0.44) SIRT6HTR6AGXTHTR3AKDM4E
SCHEMBL13243994 0.80 SIRT6 (0.63) SIRT6HTR6HTR3ADRD2DRD3
SCHEMBL22652120 0.79 GAA (0.58) SIRT6HTR6AGXTHTR3AKDM4E
SCHEMBL30602337 0.79 AGXT (0.44) SIRT6HTR6AGXTHTR3AKDM4E
SCHEMBL1911875 0.78 SIRT6 (0.60) SIRT6HTR6HTR3ADRD2DRD3
SCHEMBL438444 0.76 MAPT (0.63) SIRT6HTR6HTR3ADRD2DRD3
SCHEMBL24992445 0.76 SIRT6 (0.58) SIRT6HTR6HTR3ADRD2DRD3
SCHEMBL14145814 0.76 SIRT6 (0.58) SIRT6HTR6HTR3ADRD2DRD3
SCHEMBL24783778 0.76 SIRT6 (0.58) SIRT6HTR6HTR3ADRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11344553-B2 Substituted pyrazolopyrimidines useful as kinases inhibitors TELIGENE LTD. (CN) 2022-05-31 US disclosed
US-20210315899-A1 SUBSTITUTED PYRAZOLOPYRIMIDINES USEFUL AS KINASES INHIBITORS TELIGENE LTD. (CN) 2021-10-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210315899-A1 SUBSTITUTED PYRAZOLOPYRIMIDINES USEFUL AS KINASES INHIBITORS MAP3K20, MAP3K6, MAP3K8 SIRT6 2006/4885HTR6 3762/4885AGXT 2738/4885
US-11344553-B2 Substituted pyrazolopyrimidines useful as kinases inhibitors MAP3K20, PRKDC, MAP3K6 SIRT6 1971/4885HTR6 3465/4885AGXT 2596/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.