SCHEMBL2392289

SCHEMBL2392289

CCOC(=O)/C=C/c1cccc(OS(=O)(=O)C(F)(F)F)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.52
ALDH1A1 P00352 4/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
TTR P02766 1/20 0.50
DPP4 P27487 1/20 0.50
CYP3A4 P08684 1/20 0.48
PTGS2 P35354 1/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
MAOB P27338 1/20 0.46
MAPT P10636 2/20 0.46
DRD2 P14416 1/20 0.45
DRD3 P35462 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
BACE1 P56817 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27537154 1.00 KDM4E (0.52) KDM4EALDH1A1SMN1; SMN2TTRDPP4
SCHEMBL27519791 0.86 DRD2 (0.49) KDM4EALDH1A1SMN1; SMN2TTRPTGS2
SCHEMBL1895094 0.84 MAPT (0.53) KDM4EALDH1A1SMN1; SMN2TTRDPP4
SCHEMBL1895095 0.84 MAPT (0.53) KDM4EALDH1A1SMN1; SMN2TTRDPP4
SCHEMBL6022915 0.83 KDM4E (0.57) KDM4EALDH1A1SMN1; SMN2PTGS2MAOB
SCHEMBL6022919 0.83 KDM4E (0.57) KDM4EALDH1A1SMN1; SMN2PTGS2MAOB
SCHEMBL2390189 0.82 TTR (0.52) TTRDPP4CYP3A4PTGS2CA12
SCHEMBL5209596 0.81 TTR (0.51) KDM4EALDH1A1SMN1; SMN2TTRDPP4
SCHEMBL2389633 0.81 CYP3A4 (0.48) TTRDPP4CYP3A4PTGS2CA12
SCHEMBL9643718 0.81 ALOX5 (0.62) KDM4EALDH1A1SMN1; SMN2TTRDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE42700-E1 Induction of apoptosis in cancer cells SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2011-09-13 US disclosed
CN-1282243-A Pharmaceutical composition containing anilide derivative for antagonizing CCR5 TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-01-31 CN disclosed