SCHEMBL23926470

SCHEMBL23926470

Cc1cnc(C(=O)Nc2nc3ccc([N+](=O)[O-])cc3s2)cn1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.66
DYRK1A Q13627 1/20 0.66
NPC1 O15118 4/20 0.63
RAB9A P51151 4/20 0.63
MCL1 Q07820 1/20 0.63
KMT2A Q03164 4/20 0.62
CACNA1B Q00975 1/20 0.61
APBA1 Q02410 1/20 0.61
ALDH1A1 P00352 6/20 0.61
SMN1; SMN2 Q16637 4/20 0.61
LMNA P02545 2/20 0.61
MEN1 O00255 3/20 0.60
POLB P06746 1/20 0.60
STAT1 P42224 1/20 0.60
RXFP1 Q9HBX9 1/20 0.60
MMP13 P45452 1/20 0.59
NOD2 Q9HC29 1/20 0.58
CXCR2 P25025 1/20 0.58
ACP1 P24666 1/20 0.57
HTT P42858 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31219382 1.00 MAPT (0.66) MAPTDYRK1ANPC1RAB9AMCL1
SCHEMBL23926521 0.91 MAPT (0.58) MAPTDYRK1ANPC1RAB9AMCL1
SCHEMBL31219258 0.91 MAPT (0.58) MAPTDYRK1ANPC1RAB9AMCL1
SCHEMBL23926482 0.86 NPC1 (0.65) MAPTDYRK1ANPC1RAB9AMCL1
SCHEMBL23926494 0.85 MAPT (0.70) MAPTNPC1RAB9AKMT2AALDH1A1
SCHEMBL2486624 0.85 MAPT (0.62) MAPTDYRK1ANPC1RAB9AMCL1
SCHEMBL22130263 0.85 NPC1 (0.69) MAPTDYRK1ANPC1RAB9AMCL1
SCHEMBL31219300 0.85 NPC1 (0.69) MAPTDYRK1ANPC1RAB9AMCL1
SCHEMBL25382210 0.83 MAPT (0.51) MAPTDYRK1ANPC1RAB9AMCL1
SCHEMBL23926486 0.83 NPC1 (0.71) MAPTDYRK1ANPC1RAB9AMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12590071-B2 Hydrazone derivative in which terminal amine group is substituted with aryl group or heteroaryl group, and use thereof KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2026-03-31 US disclosed
US-20220396553-A1 NOVEL HYDRAZONE DERIVATIVE IN WHICH TERMINAL AMINE GROUP IS SUBSTITUTED WITH ARYL GROUP OR HETEROARYL GROUP, AND USE THEREOF KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2022-12-15 US disclosed
CN-113727972-A Novel hydrazone derivatives in which terminal amino group is substituted with aryl or heteroaryl group, and use thereof 韩国科学技术研究院 2021-11-30 CN disclosed
EP-3901139-A1 NOVEL HYDRAZONE DERIVATIVE WITH ARYL OR HETEROARYL GROUP SUBSTITUTED AT TERMINAL AMINE GROUP THEREOF AND USE THEREOF Korea Institute of Science and Technology (KR) 2021-10-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12590071-B2 Hydrazone derivative in which terminal amine group is substituted with aryl group or heteroaryl group, and use thereof ABL1, TH, CYP3A43 MAPT 3633/4885DYRK1A 1279/4885NPC1 1264/4885
US-20220396553-A1 NOVEL HYDRAZONE DERIVATIVE IN WHICH TERMINAL AMINE GROUP IS SUBSTITUTED WITH ARYL GROUP OR HETEROARYL GROUP, AND USE THEREOF AANAT, NAT1, HNMT MAPT 3061/4885DYRK1A 3095/4885NPC1 3755/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.