SCHEMBL23937757

SCHEMBL23937757

CNS(=O)(=O)c1cc2c(ccn2C)c(O)n1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.35
FTO Q9C0B1 1/20 0.33
CYP2A6 P11509 1/20 0.33
SIRT6 Q8N6T7 1/20 0.32
RORC P51449 2/20 0.32
PFKFB3 Q16875 1/20 0.32
TSHR P16473 1/20 0.31
KDM4E B2RXH2 1/20 0.31
TRPM8 Q7Z2W7 1/20 0.31
LMNA P02545 2/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20674252 0.82 PIK3CB (0.34) CYP2A6RORCKDM4ETRPM8
SCHEMBL20674060 0.82
SCHEMBL20674087 0.78 CCR4 (0.34) FTO
SCHEMBL23937755 0.77 FTO (0.36) PKMFTOPFKFB3TSHRLMNA
SCHEMBL20674256 0.77 TSHR (0.32) TSHR
SCHEMBL23937759 0.74 TSHR (0.43) PKMFTOSIRT6RORCTSHR
SCHEMBL23937850 0.72 BAZ2B (0.40) PKMTSHRKDM4ELMNA
SCHEMBL23937743 0.72 FTO (0.34) FTOLMNA
SCHEMBL21440750 0.70
SCHEMBL20674250 0.69 LCK (0.38) KDM4ELMNASYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed