SCHEMBL23937870

SCHEMBL23937870

CCc1nc(C#N)n2ccccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 0.38
ALDH1A1 P00352 10/20 0.38
HPGD P15428 6/20 0.38
GAA P10253 4/20 0.38
GLA P06280 2/20 0.38
KMT2A Q03164 5/20 0.38
MAPT P10636 4/20 0.38
MEN1 O00255 4/20 0.38
LMNA P02545 4/20 0.36
MAPK1 P28482 3/20 0.36
HSD17B10 Q99714 2/20 0.36
PTPN1 P18031 2/20 0.36
L3MBTL1 Q9Y468 3/20 0.35
HTT P42858 2/20 0.35
NCOA3 Q9Y6Q9 2/20 0.35
PABPC1 P11940 1/20 0.35
CASP3 P42574 1/20 0.35
NCOA1 Q15788 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20142239 0.78 PTPN1 (0.41) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL20139203 0.77 PTPN1 (0.43) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL20141604 0.77 AR (0.38) HPGDGAAKMT2AMAPTMEN1
SCHEMBL18032960 0.76 DRD4 (0.41) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL20674556 0.75 KDM4E (0.43) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL2743125 0.73 CNR2 (0.55) PTPN2
SCHEMBL20927196 0.72 HTR4 (0.44) KDM4EALDH1A1KMT2AMAPTMEN1
SCHEMBL14627434 0.72 ALDH1A1 (0.40) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL25539525 0.70 CNR2 (0.50) KDM4EALDH1A1HPGDGAAKMT2A
SCHEMBL14629325 0.69 KDM4E (0.46) KDM4EALDH1A1HPGDGAAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed