SCHEMBL23937885

SCHEMBL23937885

On1nc(C(F)(F)F)c2c1CCC2

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.51
TSHR P16473 3/20 0.50
GAA P10253 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
TDP1 Q9NUW8 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HTT P42858 1/20 0.46
GRIA2 P42262 5/20 0.44
CYP1A2 P05177 4/20 0.44
CYP2C9 P11712 1/20 0.44
MAPT P10636 3/20 0.43
THRB P10828 1/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2D6 P10635 3/20 0.42
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20631707 0.80 GRIA2 (0.41) LMNATSHRGAANPSR1TDP1
SCHEMBL20631124 0.76 LMNA (0.36) LMNATSHRGAANPSR1ALDH1A1
SCHEMBL21959600 0.75 LMNA (0.34) LMNATSHRGAANPSR1ALDH1A1
SCHEMBL20631145 0.74 LMNA (0.30) LMNA
SCHEMBL20430159 0.73 LMNA (0.51) LMNATSHRGAANPSR1ALDH1A1
SCHEMBL14401055 0.73 LMNA (0.55) LMNATSHRGAANPSR1TDP1
SCHEMBL20371630 0.73 TDP1 (0.59) LMNATSHRGAANPSR1TDP1
SCHEMBL15730538 0.72 LMNA (0.56) LMNATSHRGAANPSR1TDP1
SCHEMBL17616497 0.70 LMNA (0.49) LMNATSHRGAANPSR1TDP1
SCHEMBL20631148 0.69 PTGS2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed