SCHEMBL23938540

SCHEMBL23938540

C=CCc1ccc(C(F)(F)F)cc1CC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
ESR1 P03372 2/20 0.36
ESR2 Q92731 2/20 0.36
CES2 O00748 1/20 0.36
IDO1 P14902 2/20 0.36
DAO P14920 1/20 0.35
DCTPP1 Q9H773 1/20 0.35
PDE2A O00408 1/20 0.35
POLQ O75417 3/20 0.34
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
TGM2 P21980 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
SRD5A2 P31213 1/20 0.33
HTR2A P28223 1/20 0.33
SLC6A4 P31645 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15133743 0.83 ESR1 (0.44) CYP3A4CYP2D6ESR1ESR2CES2
SCHEMBL20751779 0.81 PDE2A (0.38) CYP3A4CYP2D6CES2IDO1DAO
SCHEMBL9797321 0.81 CES2 (0.37) CYP3A4CYP2D6CES2IDO1DAO
SCHEMBL18682072 0.78 ESR1 (0.40) CYP3A4CYP2D6ESR1ESR2CES2
SCHEMBL3683402 0.78 POLB (0.38) CYP3A4CYP2D6CES2IDO1DCTPP1
SCHEMBL16950844 0.77 PDE2A (0.39) ESR1ESR2CES2IDO1DAO
SCHEMBL18587153 0.77 IDO1 (0.37) CYP3A4CYP2D6CES2IDO1DCTPP1
SCHEMBL18586382 0.77 IDO1 (0.40) CYP3A4CYP2D6IDO1GABRA1GABRB2
SCHEMBL1986356 0.77 GABRA1 (0.46) CES2IDO1GABRA1GABRB2
SCHEMBL3678271 0.77 IDO1 (0.37) CYP3A4CYP2D6CES2IDO1PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3297438-B1 CCR2 MODULATORS CHEMOCENTRYX INC (US) 2021-10-20 EP disclosed