SCHEMBL23938744

SCHEMBL23938744

COc1ccc(Cn2ncc3cc(Br)cc(C)c32)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 10/20 0.46
MCHR1 Q99705 1/20 0.44
PDE1A P54750 3/20 0.43
PDE1B Q01064 3/20 0.43
PDE1C Q14123 3/20 0.43
PKM P14618 1/20 0.43
PKLR P30613 1/20 0.43
DCTPP1 Q9H773 1/20 0.42
IDO1 P14902 1/20 0.41
P2RX7 Q99572 1/20 0.41
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
BRD4 O60885 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALOX15 P16050 1/20 0.40
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18301358 0.86 NPBWR1 (0.44) NPBWR1MCHR1PDE1APDE1BPDE1C
SCHEMBL29161724 0.84 TSHR (0.50) PKMPKLRP2RX7ALDH1A1MAPT
SCHEMBL759935 0.81 NPBWR1 (0.44) NPBWR1MCHR1PKMPKLRALDH1A1
SCHEMBL530059 0.79 IDO1 (0.47) NPBWR1MCHR1PDE1APDE1BPDE1C
SCHEMBL2961568 0.78 PDE1B (0.52) NPBWR1MCHR1PDE1APDE1BPDE1C
SCHEMBL29433484 0.76 BRD4 (0.53) NPBWR1MCHR1PDE1APDE1BPDE1C
SCHEMBL27242636 0.76 NPBWR1 (0.47) NPBWR1MCHR1PDE1APDE1BPDE1C
SCHEMBL20176889 0.76 NPBWR1 (0.47) NPBWR1MCHR1PDE1APDE1BPDE1C
SCHEMBL5091051 0.76 BRD4 (0.53) NPBWR1MCHR1PDE1APDE1BPDE1C
SCHEMBL24785427 0.76 NPBWR1 (0.43) NPBWR1MCHR1P2RX7MAPTBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3307733-B1 MANNOSE DERIVATIVES FOR TREATING BACTERIAL INFECTIONS VERTEX PHARMA (US) 2021-10-20 EP disclosed