SCHEMBL23948298

SCHEMBL23948298

COc1cnccc1-c1cnn(-c2cnn3ccc(=O)[nH]c23)c1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MELK Q14680 11/20 0.47
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
GRM4 Q14833 1/20 0.35
PDGFRA P16234 1/20 0.34
FLT3 P36888 1/20 0.34
HASPIN Q8TF76 1/20 0.34
HAVCR2 Q8TDQ0 1/20 0.34
PLAT P00750 2/20 0.33
CREBBP Q92793 1/20 0.33
AAK1 Q2M2I8 2/20 0.32
BUB1 O43683 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23948447 0.92 MELK (0.38) MELKGRM4FLT3PLATCREBBP
SCHEMBL26306170 0.87 PLAT (0.42) PLATCREBBP
SCHEMBL23948455 0.84 MELK (0.43) MELKGRM4
SCHEMBL23948322 0.81 MELK (0.40) MELKPLAT
SCHEMBL23948445 0.80 BTK (0.40) GRM4CREBBPAAK1
SCHEMBL23948444 0.78 KDR (0.31) FLT3PLAT
SCHEMBL23948328 0.78 ABL1 (0.38) PLAT
SCHEMBL23948294 0.78 CYP11B1 (0.38) PLAT
SCHEMBL26309079 0.77 HCAR1 (0.36) PLAT
SCHEMBL23947949 0.77 PDE10A (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230242536-A1 METHODS FOR PREPARING TYROSINE RECEPTOR KINASE INHIBITORS PYRAMID BIOSCIENCES, INC. 2023-08-03 US disclosed
WO-2021211882-A1 METHODS FOR PREPARING TYROSINE RECEPTOR KINASE INHIBITORS PYRAMID BIOSCIENCES, INC. (US) 2021-10-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242536-A1 METHODS FOR PREPARING TYROSINE RECEPTOR KINASE INHIBITORS LTK, FRK, LCK MELK 151/4885CCNC 1675/4885CDK8 207/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.