SCHEMBL23948447

SCHEMBL23948447

COc1ccncc1-c1cnn(-c2cnn3ccc(=O)[nH]c23)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MELK Q14680 2/20 0.38
GSK3B P49841 6/20 0.33
IKBKB O14920 1/20 0.33
CHUK O15111 1/20 0.33
CREBBP Q92793 1/20 0.33
LRRK2 Q5S007 1/20 0.33
GRM4 Q14833 1/20 0.33
JAK2 O60674 1/20 0.32
CDK2 P24941 1/20 0.32
KDR P35968 1/20 0.32
FLT3 P36888 1/20 0.32
SYK P43405 1/20 0.32
PIK3CG P48736 1/20 0.32
MAPK10 P53779 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
CCNT1 O60563 1/20 0.32
CDK9 P50750 1/20 0.32
PLAT P00750 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23948298 0.92 MELK (0.47) MELKCREBBPGRM4FLT3PLAT
SCHEMBL26306170 0.87 PLAT (0.42) CREBBPPLATHCAR1
SCHEMBL23948455 0.82 MELK (0.43) MELKGSK3BGRM4CDK2IRAK4
SCHEMBL23948322 0.81 MELK (0.40) MELKKDRPLATHCAR1
SCHEMBL23948445 0.80 BTK (0.40) CREBBPGRM4
SCHEMBL23948444 0.78 KDR (0.31) GSK3BCDK2KDRFLT3PLAT
SCHEMBL23948328 0.78 ABL1 (0.38) PLATCYP11B2
SCHEMBL23948294 0.78 CYP11B1 (0.38) PIK3CGPLATCYP11B2
SCHEMBL26309079 0.77 HCAR1 (0.36) IRAK4PLATHCAR1
SCHEMBL23947949 0.77 PDE10A (0.34) HCAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230242536-A1 METHODS FOR PREPARING TYROSINE RECEPTOR KINASE INHIBITORS PYRAMID BIOSCIENCES, INC. 2023-08-03 US disclosed
US-20230242536-A1 METHODS FOR PREPARING TYROSINE RECEPTOR KINASE INHIBITORS PYRAMID BIOSCIENCES, INC. 2023-08-03 US disclosed
WO-2021211882-A1 METHODS FOR PREPARING TYROSINE RECEPTOR KINASE INHIBITORS PYRAMID BIOSCIENCES, INC. (US) 2021-10-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242536-A1 METHODS FOR PREPARING TYROSINE RECEPTOR KINASE INHIBITORS LTK, FRK, LCK MELK 151/4885GSK3B 1015/4885IKBKB 588/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.