SCHEMBL23950265

SCHEMBL23950265

O=c1c2cc(-c3ccc(C(F)(F)F)cc3)nc(-c3cccnc3)c2ncn1CCCO

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.39
TOP1 P11387 2/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
PIM1 P11309 1/20 0.38
MAPT P10636 2/20 0.37
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
GSK3B P49841 2/20 0.37
MAP4K4 O95819 2/20 0.37
MAPK9 P45984 2/20 0.37
CSNK1A1 P48729 2/20 0.37
CSNK1D P48730 2/20 0.37
MAP4K5 Q9Y4K4 2/20 0.37
PRKD3 O94806 1/20 0.37
FRK P42685 1/20 0.37
PRKD2 Q9BZL6 1/20 0.37
CCNB2 O95067 1/20 0.36
CDK1 P06493 1/20 0.36
CCNB1 P14635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23950293 0.87 PTGS2 (0.42) EGLN1TOP1PIM1PTGS1PTGS2
SCHEMBL23950296 0.87 GRM2 (0.38) EGLN1TOP1PIM1MAPTPTGS1
SCHEMBL23950768 0.86 EGLN1 (0.38) EGLN1TOP1PIM1MAPTPTGS1
SCHEMBL23950264 0.86 EGLN1 (0.38) EGLN1TOP1PIM1MAPTPTGS1
SCHEMBL23390502 0.86 SMN1; SMN2 (0.38) EGLN1TOP1PIM1MAPTPTGS1
SCHEMBL23951123 0.85 PIM1 (0.37) EGLN1TOP1PIM1MAPTPTGS1
SCHEMBL30102064 0.85 PIM1 (0.37) EGLN1TOP1PIM1MAPTPTGS1
SCHEMBL26294729 0.85 HSP90AA1 (0.39) PIM1PTGS1PTGS2GRM2
SCHEMBL23950531 0.84 PIM1 (0.41) EGLN1TOP1PIM1MAPTPTGS1
SCHEMBL23390067 0.83 AHR (0.45) NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021210970-A1 PYRIDOPYRIMIDINONE DERIVATIVES AND THEIR USE AS ARYL HYDROCARBON RECEPTOR MODULATORS DONG-A ST CO., LTD. (KR) 2021-10-21 WO disclosed