SCHEMBL23958146

SCHEMBL23958146

Cc1cc(Nc2nc3ccc(F)cc3c(=O)n2-c2ccccc2)ccn1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 2/20 0.45
IDO2 Q6ZQW0 2/20 0.45
POLB P06746 1/20 0.44
PIK3CD O00329 1/20 0.42
PIK3CG P48736 1/20 0.42
PIK3C3 Q8NEB9 1/20 0.42
IDO1 P14902 1/20 0.41
TGFBR1 P36897 1/20 0.41
KCNH2 Q12809 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GLA P06280 1/20 0.40
MAT2A P31153 1/20 0.39
PIK3CB P42338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23931388 0.89 TDO2 (0.44) TDO2IDO2POLBPIK3CDPIK3CG
SCHEMBL30103205 0.89 TDO2 (0.44) TDO2IDO2POLBPIK3CDPIK3CG
SCHEMBL23958170 0.87 POLB (0.42) TDO2IDO2POLBPIK3CDPIK3CG
SCHEMBL23958281 0.86 TDO2 (0.46) TDO2IDO2POLBPIK3CDPIK3CG
SCHEMBL23958194 0.85 TDO2 (0.46) TDO2IDO2POLBPIK3CDPIK3CG
SCHEMBL29623155 0.85 TDO2 (0.50) TDO2IDO2POLBPIK3CDPIK3CG
SCHEMBL23045334 0.85 TDO2 (0.50) TDO2IDO2POLBPIK3CDPIK3CG
SCHEMBL24110965 0.83 POLB (0.49) TDO2IDO2POLBPIK3CDPIK3CG
SCHEMBL24110956 0.83 TDO2 (0.44) TDO2IDO2POLBPIK3CDPIK3CG
SCHEMBL24111048 0.82 TDO2 (0.46) TDO2IDO2POLBPIK3CDPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210387967-A1 2-HETEROARYL AMINOQUINAZOLINONE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2021-12-16 US disclosed
WO-2021215537-A1 2-HETEROARYLAMINOQUINAZOLINONE DERIVATIVE 大日本住友製薬株式会社 (JP) 2021-10-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210387967-A1 2-HETEROARYL AMINOQUINAZOLINONE DERIVATIVE CRKL, CLIC4, CLIC1 TDO2 1621/4885IDO2 443/4885POLB 4618/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.