SCHEMBL23958630

SCHEMBL23958630

COC(=O)c1cc(/C=C(\N)C(F)F)c(N)c(OC)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.40
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
LMNA P02545 2/20 0.38
ATM Q13315 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KDM4E B2RXH2 6/20 0.38
POLB P06746 3/20 0.38
CNR2 P34972 1/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP3A4 P08684 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
USP2 O75604 1/20 0.35
ERN1 O75460 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958934 0.88 CA12 (0.44) MAPTLMNAKDM4ECNR2ALDH1A1
SCHEMBL23958596 0.83 MAPT (0.44) MAPTKMT2AMEN1LMNAATM
SCHEMBL23958822 0.78 KDM4E (0.39) MAPTKMT2AMEN1LMNAATM
SCHEMBL10683847 0.76 KDM4E (0.53) MAPTKMT2AMEN1LMNAATM
SCHEMBL23958829 0.75 NOTUM (0.38) MAPTKMT2AMEN1LMNAATM
SCHEMBL16545267 0.74 KDM4E (0.40) MAPTKMT2AMEN1LMNAATM
SCHEMBL23958621 0.72 PDE4B (0.38)
SCHEMBL18031417 0.72 KDM4E (0.53) MAPTKMT2ALMNAATMNPSR1
SCHEMBL30418756 0.72 KDM4E (0.53) MAPTKMT2ALMNAATMNPSR1
SCHEMBL23905892 0.70 CNR2 (0.49) MAPTKMT2AMEN1LMNAATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed