SCHEMBL23958700

SCHEMBL23958700

COc1cc(C(=O)NCC(c2nc(-c3ccc(F)cc3)c(F)c(C(C)(C)O)c2F)C2CC2)cc2cc(C3CC3)nnc12

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
ROCK2 O75116 10/20 0.33
ROCK1 Q13464 10/20 0.33
ALDH1A1 P00352 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TLR9 Q9NR96 1/20 0.32
TLR8 Q9NR97 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
KCNH2 Q12809 1/20 0.31
MAPT P10636 1/20 0.31
ACSS2 Q9NR19 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25282615 0.84 ROCK2 (0.33) LMNATP53ROCK2ROCK1MAPT
SCHEMBL25687434 0.84 ROCK2 (0.33) LMNATP53ROCK2ROCK1MAPT
SCHEMBL25697480 0.83
SCHEMBL23958792 0.80 CFTR (0.33) LMNATP53ROCK2ROCK1ALDH1A1
SCHEMBL23958806 0.80 CFTR (0.34) LMNATP53ROCK2ROCK1ALDH1A1
SCHEMBL23958703 0.79 CFTR (0.32) LMNATP53ROCK2ROCK1ALDH1A1
SCHEMBL30007492 0.78 CFTR (0.34) ROCK2ROCK1SMN1; SMN2KCNH2MAPT
SCHEMBL30007120 0.78 CFTR (0.36) ROCK2ROCK1ALDH1A1SMN1; SMN2KCNH2
SCHEMBL28909115 0.78 CFTR (0.36) ROCK2ROCK1ALDH1A1SMN1; SMN2KCNH2
SCHEMBL25282974 0.78 CFTR (0.34) ROCK2ROCK1SMN1; SMN2KCNH2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed