SCHEMBL23958703

SCHEMBL23958703

COc1cc(C(=O)NCC(c2nc(-c3ccc(F)cc3)c(F)c(C(C)(C)O)c2F)C2CC2)cc(/C=C(\N)C2CC2)c1N

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.32
MAPT P10636 3/20 0.32
ALDH1A1 P00352 3/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TLR9 Q9NR96 1/20 0.31
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
POLB P06746 2/20 0.31
NAMPT P43490 1/20 0.31
KMT2A Q03164 1/20 0.31
KCNH2 Q12809 1/20 0.31
ACKR3 P25106 1/20 0.30
KDM4E B2RXH2 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958792 0.93 CFTR (0.33) CFTRMAPTALDH1A1LMNATP53
SCHEMBL23958779 0.84 MAPT (0.33) MAPTALDH1A1LMNATP53SMN1; SMN2
SCHEMBL23958700 0.79 LMNA (0.34) MAPTALDH1A1LMNATP53SMN1; SMN2
SCHEMBL23958782 0.78 CFTR (0.35) CFTRMAPTALDH1A1LMNATP53
SCHEMBL23958894 0.77 CFTR (0.34) CFTRMAPTALDH1A1LMNATP53
SCHEMBL23958775 0.75 ADRA1D (0.36) CFTRMAPTALDH1A1SMN1; SMN2ROCK2
SCHEMBL23958976 0.75 KDM4E (0.31) CFTRMAPTALDH1A1POLBKDM4E
SCHEMBL23958744 0.74 SCN9A (0.32) MAPTLMNANAMPTKDM4E
SCHEMBL23958812 0.73 CFTR (0.38) CFTRMAPTALDH1A1ROCK2ROCK1
SCHEMBL23958860 0.71 RPS6KB1 (0.33) CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed