SCHEMBL23959077

SCHEMBL23959077

C#CCCC1(c2ccccc2C)C(=O)N(C(=O)OC(C)(C)C)c2ccc(F)cc21

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 7/20 0.39
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
BCHE P06276 1/20 0.35
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PKM P14618 1/20 0.31
KCNQ4 P56696 1/20 0.30
KCNQ5 Q9NR82 1/20 0.30
IDO1 P14902 1/20 0.30
TDO2 P48775 1/20 0.30
IDO2 Q6ZQW0 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TP53 P04637 1/20 0.30
ADAMTS5 Q9UNA0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23959074 0.83 CASP1 (0.38) CASP1PDE4APDE4BPDE4CPDE4D
SCHEMBL23959043 0.76 PDE4A (0.38) CASP1PDE4APDE4BPDE4CPDE4D
SCHEMBL23959073 0.72 ALDH1A1 (0.38) CASP1PDE4APDE4BPDE4CPDE4D
SCHEMBL23959063 0.72 ALDH1A1 (0.38) CASP1PDE4APDE4BPDE4CPDE4D
SCHEMBL31526042 0.72 CASP1 (0.40) CASP1BCHEIDO1TDO2IDO2
SCHEMBL18025794 0.71 CASP1 (0.42) CASP1PDE4APDE4BPDE4CPDE4D
SCHEMBL23959079 0.69 CASP1 (0.37) CASP1PDE4APDE4BPDE4CPDE4D
SCHEMBL30594659 0.69 BCHE (0.44) CASP1PDE4APDE4BPDE4CPDE4D
SCHEMBL23959115 0.68 PDE4A (0.41) CASP1PDE4APDE4BPDE4CPDE4D
SCHEMBL23959127 0.68 PDE4A (0.41) CASP1PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021212974-A1 RACEMIC AND CHIRAL 3-(2,3-BUTADIENYL)OXYINDOLINONE COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 复旦大学 (CN) 2021-10-28 WO disclosed