SCHEMBL23960283

SCHEMBL23960283

CC(C)(C)OC(=O)Nc1c(Cl)csc1CF

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.41
LCK P06239 6/20 0.39
METAP1 P53582 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
MAPKAPK2 P49137 2/20 0.34
GAA P10253 1/20 0.33
APLNR P35414 1/20 0.33
CYP17A1 P05093 1/20 0.33
STK17B O94768 1/20 0.33
STK17A Q9UEE5 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23960284 0.82 ATR (0.43) ATRLCKMETAP1PI4KBMAPKAPK2
SCHEMBL23960286 0.80 ATR (0.41) ATRLCKMETAP1PI4KBCA12
SCHEMBL23960289 0.79 ATR (0.40) ATRLCKGAAAPLNRCA12
SCHEMBL23960254 0.79 ATR (0.40) ATRLCKMETAP1PI4KBMAPKAPK2
SCHEMBL25170234 0.78 KMT2A (0.43) ATRLCKGAACA12CA1
SCHEMBL25170226 0.78 ATR (0.42) ATRLCKPI4KBGAACA12
SCHEMBL25168106 0.77 ATR (0.50) ATRLCKCA12CA1CA2
SCHEMBL23960260 0.74 ATR (0.43) ATRLCKMETAP1PI4KBCYP17A1
SCHEMBL25434214 0.73 ATR (0.41) ATRLCKMAPKAPK2CA12CA1
SCHEMBL22774841 0.72 ATR (0.38) ATRLCKMETAP1PI4KBCYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230348453-A1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF IOMX THERAPEUTICS AG (DE) 2023-11-02 US disclosed
US-20230192701-A1 BICYCLIC KINASE INHIBITORS AND USES THEREOF IOMX THERAPEUTICS AG (DE) 2023-06-22 US disclosed
WO-2021219731-A2 BICYCLIC KINASE INHIBITORS AND USES THEREOF IOMX THERAPEUTICS AG (DE) 2021-11-04 WO disclosed
WO-2021214117-A1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF IOMX THERAPEUTICS AG (DE) 2021-10-28 WO disclosed
EP-3901151-A1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF iOmx Therapeutics AG (DE) 2021-10-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230348453-A1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF ABL1, PRKDC, PRKACA ATR 1763/4885LCK 72/4885METAP1 1796/4885
US-20230192701-A1 BICYCLIC KINASE INHIBITORS AND USES THEREOF MITF, PRKDC, PRKACA ATR 1283/4885LCK 122/4885METAP1 1572/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.