SCHEMBL23960254

SCHEMBL23960254

CC(C)(C)OC(=O)Nc1c(CF)csc1Cl

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.40
LCK P06239 5/20 0.36
PI4KB Q9UBF8 1/20 0.34
GAA P10253 1/20 0.33
CYP17A1 P05093 1/20 0.33
APLNR P35414 1/20 0.33
CTSL P07711 1/20 0.32
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
MAPKAPK2 P49137 1/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 1/20 0.32
METAP1 P53582 1/20 0.32
CA12 O43570 1/20 0.32
CA9 Q16790 1/20 0.32
PSMB8 P28062 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23960309 0.87 ATR (0.41) ATRLCKPI4KBGAACYP17A1
SCHEMBL23987746 0.82 ATR (0.32) ATRLCK
SCHEMBL23960260 0.81 ATR (0.43) ATRLCKPI4KBCYP17A1CA1
SCHEMBL3043609 0.80 ATR (0.44) ATRLCKPI4KBCA1CA12
SCHEMBL23960262 0.79 LMNA (0.42) ATRLCKPI4KBCA1CA2
SCHEMBL23960283 0.79 ATR (0.41) ATRLCKPI4KBGAACYP17A1
SCHEMBL23960257 0.78 ATR (0.40) ATRLCKPI4KBAPLNRCA1
SCHEMBL23927263 0.77 KEAP1 (0.30)
SCHEMBL23960341 0.76 ATR (0.44) ATRLCKPI4KBCYP17A1CA1
SCHEMBL23927246 0.76 ATR (0.56) ATRLCKCA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3901151-B1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF IOMX THERAPEUTICS AG (DE) 2026-04-01 EP disclosed
US-20250296928-A1 A SYNTHESIS SCHEME AND PROCEDURES FOR PREPARING A SIK3 INHIBITOR AND INTERMEDIATES THEREOF IOMX THERAPEUTICS AG (DE) 2025-09-25 US disclosed
CN-118369321-A Synthetic schemes and procedures for preparing SIK3 inhibitors and intermediates thereof 艾奥麦克斯治疗公司 2024-07-19 CN disclosed
US-20230348453-A1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF IOMX THERAPEUTICS AG (DE) 2023-11-02 US disclosed
US-20230348453-A1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF IOMX THERAPEUTICS AG (DE) 2023-11-02 US disclosed
US-20230348453-A1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF IOMX THERAPEUTICS AG (DE) 2023-11-02 US disclosed
US-20230192701-A1 BICYCLIC KINASE INHIBITORS AND USES THEREOF IOMX THERAPEUTICS AG (DE) 2023-06-22 US disclosed
WO-2023067021-A1 A SYNTHESIS SCHEME AND PROCEDURES FOR PREPARING A SIK3 INHIBITOR AND INTERMEDIATES THEREOF IOMX THERAPEUTICS AG (DE) 2023-04-27 WO disclosed
EP-4139305-A1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF iOmx Therapeutics AG (DE) 2023-03-01 EP disclosed
CN-115667255-A Halogenated heteroaryl and other heterocyclic kinase inhibitors and uses thereof 艾欧麦克斯治疗股份公司 2023-01-31 CN disclosed
WO-2021219731-A2 BICYCLIC KINASE INHIBITORS AND USES THEREOF IOMX THERAPEUTICS AG (DE) 2021-11-04 WO disclosed
WO-2021214117-A1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF IOMX THERAPEUTICS AG (DE) 2021-10-28 WO disclosed
EP-3901151-A1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF iOmx Therapeutics AG (DE) 2021-10-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230348453-A1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF ABL1, PRKDC, PRKACA ATR 1763/4885LCK 72/4885PI4KB 758/4885
US-20230192701-A1 BICYCLIC KINASE INHIBITORS AND USES THEREOF MITF, PRKDC, PRKACA ATR 1283/4885LCK 122/4885PI4KB 853/4885
US-20250296928-A1 A SYNTHESIS SCHEME AND PROCEDURES FOR PREPARING A SIK3 INHIBITOR AND INTERMEDIATES THEREOF SIK3, SIK1, SIK2 ATR 615/4885LCK 769/4885PI4KB 95/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.