SCHEMBL2396614

SCHEMBL2396614

CSc1ccc(OC(F)(F)[C@H](NC(CS)C(=O)O)c2ccc(F)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 6/20 0.42
CTSS P25774 3/20 0.42
CTSK P43235 3/20 0.42
CTSB P07858 2/20 0.42
LMNA P02545 2/20 0.38
GAA P10253 1/20 0.38
ACE P12821 5/20 0.38
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CRHBP P24387 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
CRHR2 Q13324 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MME P08473 3/20 0.36
NR3C1 P04150 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2396618 1.00 CTSL (0.42) CTSLCTSSCTSKCTSBLMNA
SCHEMBL2398750 0.83 KIF11 (0.47) CTSLCTSSCTSKCTSB
SCHEMBL2398747 0.83 KIF11 (0.47) CTSLCTSSCTSKCTSB
SCHEMBL2401298 0.83 CTSL (0.37) CTSLCTSSCTSKCTSBLMNA
SCHEMBL1272546 0.79 CTSL (0.53) CTSLCTSSCTSKCTSBACE
SCHEMBL1272545 0.79 CTSL (0.53) CTSLCTSSCTSKCTSBACE
SCHEMBL2346160 0.77 ACE (0.39) CTSLCTSSCTSKCTSBACE
SCHEMBL2346150 0.77 ACE (0.39) CTSLCTSSCTSKCTSBACE
SCHEMBL1272477 0.75 CTSL (0.44) CTSLCTSSCTSKCTSBACE
SCHEMBL1272478 0.75 CTSL (0.44) CTSLCTSSCTSKCTSBACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8013186-B2 Haloalkyl containing compounds as cysteine protease inhibitors VIROBAY, INC. (US) 2011-09-06 US disclosed