SCHEMBL23966554

SCHEMBL23966554

CCOC(=O)Cn1nc(Cc2cc3cc(Cl)c(OCC(F)F)cc3n2COCC[C@@H](C)CC)c2ccccc2c1=O

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 10/20 0.47
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
GAA P10253 1/20 0.36
RECQL P46063 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23909043 0.91 S1PR2 (0.48) S1PR2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL23914741 0.90 S1PR2 (0.48) S1PR2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL23914758 0.83 S1PR2 (0.57) S1PR2
SCHEMBL23914760 0.82 S1PR2 (0.56) S1PR2
SCHEMBL23966562 0.81 S1PR2 (0.36) S1PR2CYP3A4CYP2C9CYP2C19NPSR1
SCHEMBL23909060 0.80 S1PR2 (0.53) S1PR2GAAMEN1KMT2A
SCHEMBL23914732 0.79 S1PR2 (0.52) S1PR2GAAMEN1KMT2A
SCHEMBL23915376 0.71 S1PR2 (0.37) S1PR2CYP3A4CYP2C9CYP2C19L3MBTL1
SCHEMBL23915377 0.70 S1PR2 (0.37) S1PR2CYP3A4CYP2C9CYP2C19L3MBTL1
SCHEMBL23908807 0.68 S1PR2 (0.72) S1PR2CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3649119-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2021-11-03 EP disclosed