SCHEMBL23966562

SCHEMBL23966562

CC[C@H](C)CCOCn1c(Cc2n[nH]c(=O)c3ccccc23)cc2cc(Cl)c(OCC(F)F)cc21

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 1/20 0.36
AR P10275 8/20 0.35
LMNA P02545 2/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PARP1 P09874 5/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23915376 0.89 S1PR2 (0.37) S1PR2ARLMNAHTTNPSR1
SCHEMBL23915377 0.88 S1PR2 (0.37) S1PR2ARLMNAHTTNPSR1
SCHEMBL23966554 0.81 S1PR2 (0.47) S1PR2NPSR1CYP3A4CYP2C9CYP2C19
SCHEMBL23914758 0.72 S1PR2 (0.57) S1PR2TSHR
SCHEMBL23914760 0.72 S1PR2 (0.56) S1PR2TSHR
SCHEMBL23909043 0.71 S1PR2 (0.48) S1PR2NPSR1CYP3A4CYP2C9CYP2C19
SCHEMBL23966811 0.71 PARP1 (0.36) ARLMNAPARP1CYP3A4CYP2C9
SCHEMBL23914741 0.71 S1PR2 (0.48) S1PR2NPSR1CYP3A4CYP2C9CYP2C19
SCHEMBL23909113 0.66 GRM2 (0.32)
SCHEMBL23915555 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3649119-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2021-11-03 EP disclosed