SCHEMBL23966557

SCHEMBL23966557

COC(=O)N1CCC(Cn2nc(CC(=O)O)c3ccccc3c2=O)CC1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.56
AKR1B1 P15121 8/20 0.50
GPR39 O43194 1/20 0.50
KMT2A Q03164 2/20 0.47
HRH1 P35367 2/20 0.47
S1PR2 O95136 2/20 0.47
POLB P06746 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
ALOX15 P16050 1/20 0.46
NPSR1 Q6W5P4 1/20 0.45
BRD4 O60885 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23966559 0.92 GPR39 (0.50) MAPTGPR39KMT2AHRH1S1PR2
SCHEMBL23966556 0.91 MAPT (0.58) MAPTAKR1B1GPR39KMT2AHRH1
SCHEMBL23913676 0.89 MAPT (0.53) MAPTAKR1B1GPR39KMT2AHRH1
SCHEMBL23915524 0.85 MAPT (0.67) MAPTAKR1B1GPR39KMT2APOLB
SCHEMBL23966558 0.85 RECQL (0.57) MAPTGPR39HRH1ALDH1A1NPSR1
SCHEMBL23915443 0.83 MAPT (0.51) MAPTAKR1B1GPR39KMT2AHRH1
SCHEMBL23915515 0.83 NPC1 (0.49) MAPTGPR39KMT2AHRH1ADRA1A
SCHEMBL23913685 0.83 MAPT (0.64) MAPTAKR1B1GPR39KMT2AHRH1
SCHEMBL23914889 0.81 RECQL (0.56) MAPTAKR1B1GPR39HRH1S1PR2
SCHEMBL23915614 0.79 GPR39 (0.62) MAPTGPR39HRH1ADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3649119-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2021-11-03 EP disclosed