SCHEMBL23966558

SCHEMBL23966558

CCOC(=O)N1CCC(Cn2nc(CC(=O)OC)c3ccccc3c2=O)CC1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.57
NPSR1 Q6W5P4 1/20 0.54
ALDH1A1 P00352 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.50
GPR39 O43194 1/20 0.48
SLC6A4 P31645 11/20 0.46
HTR2A P28223 3/20 0.46
HTR2C P28335 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HRH1 P35367 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23966559 0.93 GPR39 (0.50) RECQLNPSR1ALDH1A1SMN1; SMN2GPR39
SCHEMBL23966556 0.90 MAPT (0.58) RECQLNPSR1ALDH1A1SMN1; SMN2GPR39
SCHEMBL23915515 0.89 NPC1 (0.49) RECQLNPSR1ALDH1A1SMN1; SMN2GPR39
SCHEMBL23914889 0.88 RECQL (0.56) RECQLALDH1A1SMN1; SMN2GPR39L3MBTL1
SCHEMBL23915614 0.85 GPR39 (0.62) RECQLALDH1A1SMN1; SMN2GPR39L3MBTL1
SCHEMBL23966557 0.85 MAPT (0.56) NPSR1ALDH1A1GPR39HRH1MAPT
SCHEMBL23915513 0.83 NPC1 (0.46) RECQLNPSR1ALDH1A1SMN1; SMN2GPR39
SCHEMBL23914890 0.80 HRH1 (0.55) RECQLALDH1A1SMN1; SMN2GPR39L3MBTL1
SCHEMBL23913676 0.78 MAPT (0.53) ALDH1A1SMN1; SMN2GPR39HRH1MAPT
SCHEMBL23915623 0.78 RECQL (0.47) RECQLALDH1A1SMN1; SMN2GPR39SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3649119-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2021-11-03 EP disclosed