SCHEMBL23966573

SCHEMBL23966573

CC(C)(C)OC(=O)N1CCC(n2nc(Cc3nc4cc(OCC(F)F)c(C#N)cc4n3SF)c3ccccc3c2=O)C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 2/20 0.35
S1PR2 O95136 1/20 0.34
PIK3CD O00329 2/20 0.33
TNF P01375 2/20 0.33
LITAF Q99732 2/20 0.33
GPR119 Q8TDV5 2/20 0.32
NSD2 O96028 3/20 0.32
TBK1 Q9UHD2 3/20 0.32
PIK3CA P42336 2/20 0.32
PIK3R2 O00459 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
PIK3R5 Q8WYR1 1/20 0.32
PIK3R3 Q92569 1/20 0.32
USP30 Q70CQ3 1/20 0.32
EHMT2 Q96KQ7 1/20 0.32
PARP1 P09874 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
ADRA1A P35348 1/20 0.31
HRH1 P35367 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23909091 0.87 BTK (0.34) BTKS1PR2PIK3CDTNFLITAF
SCHEMBL23915581 0.84 S1PR2 (0.49) BTKS1PR2PIK3CDTNFLITAF
SCHEMBL23966551 0.84 S1PR2 (0.37) S1PR2
SCHEMBL23966827 0.83 S1PR2 (0.36) S1PR2PIK3CD
SCHEMBL23915420 0.81 S1PR2 (0.33) S1PR2
SCHEMBL23915477 0.79 S1PR2 (0.52) S1PR2NSD2TBK1PARP1
SCHEMBL23966578 0.77 S1PR2 (0.44) S1PR2ADRA1AHRH1ADRA1BHRH3
SCHEMBL23966577 0.77 S1PR2 (0.38) S1PR2
SCHEMBL23914857 0.76 S1PR2 (0.43) BTKS1PR2PIK3CDTNFLITAF
SCHEMBL23915604 0.75 ADRA1A (0.37) S1PR2ADRA1AHRH1ADRA1BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3649119-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2021-11-03 EP disclosed