SCHEMBL23967175

SCHEMBL23967175

COC(=O)N1CCC2(CC1)CCN(c1ccc([N+](=O)[O-])cc1)CC2

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.67
CYP2C19 P33261 3/20 0.67
MAPK1 P28482 2/20 0.67
MEN1 O00255 1/20 0.67
KMT2A Q03164 1/20 0.67
HIF1A Q16665 2/20 0.64
MAPT P10636 8/20 0.60
ALDH1A1 P00352 8/20 0.60
LMNA P02545 3/20 0.60
SMN1; SMN2 Q16637 3/20 0.60
HSD17B10 Q99714 5/20 0.55
USP2 O75604 4/20 0.55
CYP1A2 P05177 2/20 0.54
CYP2D6 P10635 1/20 0.51
TSHR P16473 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
CYP2C9 P11712 1/20 0.50
ALOX15 P16050 1/20 0.50
HTT P42858 1/20 0.50
TP53 P04637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2105411 0.88 MAPT (0.75) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL10035910 0.86 MAPT (0.80) CYP3A4CYP2C19MAPK1MEN1KMT2A
SCHEMBL21855141 0.84 MAPT (0.54) CYP2C19MAPK1MEN1KMT2AMAPT
SCHEMBL18812853 0.82 ALDH1A1 (0.64) CYP3A4CYP2C19MAPK1MEN1KMT2A
SCHEMBL23126532 0.81 CYP3A4 (0.74) CYP3A4CYP2C19MAPK1MEN1KMT2A
SCHEMBL30985057 0.81 POLB (0.51) MAPK1MEN1KMT2AMAPTALDH1A1
SCHEMBL30984960 0.80 MAPT (0.72) MAPTALDH1A1LMNASMN1; SMN2HTT
SCHEMBL13247587 0.79 SIRT6 (0.73) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL21526639 0.79 SIRT6 (0.52) CYP3A4CYP2C19MAPK1HIF1AMAPT
SCHEMBL30984732 0.79 MAPT (0.66) CYP3A4CYP2C19MAPK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3572413-B1 1,2-DIHYDRO-3H-PYRAZOLO[3,4-D]PYRIMIDIN-3-ONE DERIVATIVE AS WEE1 INHIBITOR SHIJIAZHUANG SAGACITY NEW DRUG DEV CO LTD (CN) 2021-11-03 EP disclosed