SCHEMBL23968014

SCHEMBL23968014

FC(F)(F)Oc1ccc(-n2cc(-c3ccc(N4CCSCC4)cc3)cn2)cc1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MELK Q14680 3/20 0.45
MAP4K1 Q92918 1/20 0.41
MAPKAPK2 P49137 1/20 0.40
SCN5A Q14524 7/20 0.39
KCNA5 P22460 1/20 0.38
RXRA P19793 5/20 0.38
GRIN1 Q05586 5/20 0.38
GRIN2B Q13224 5/20 0.38
FFAR4 Q5NUL3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23968071 0.89 MLYCD (0.42) MELKRXRAGRIN1GRIN2B
SCHEMBL23968199 0.84 MAPKAPK2 (0.57) MELKMAPKAPK2
SCHEMBL23968072 0.83 MELK (0.45) MELKMAP4K1MAPKAPK2RXRAGRIN1
SCHEMBL23968001 0.82 MELK (0.51) MELK
SCHEMBL23968161 0.82 S1PR1 (0.41) MELKMAP4K1
SCHEMBL23968081 0.81 MELK (0.45) MELKMAPKAPK2
SCHEMBL23968093 0.80 MAP4K4 (0.54) MELK
SCHEMBL23968106 0.79 MELK (0.43) MELK
SCHEMBL29266901 0.78 ABL1 (0.51) MELKMAPKAPK2RXRAGRIN1GRIN2B
SCHEMBL23968168 0.78 MELK (0.46) MELKMAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2021-11-03 EP disclosed