SCHEMBL23968199

SCHEMBL23968199

COc1ccc(-n2cc(-c3ccc(N4CCSCC4)cc3)cn2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 1/20 0.57
MELK Q14680 4/20 0.51
RAB9A P51151 5/20 0.47
NPC1 O15118 4/20 0.47
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
ADRB1 P08588 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
MAPT P10636 5/20 0.42
KMT2A Q03164 2/20 0.42
TGFBR1 P36897 2/20 0.41
ALDH1A1 P00352 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
FYN P06241 1/20 0.41
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23968136 0.88 MKNK1 (0.47) MAPKAPK2MELKNPC1ADRB1MAPT
SCHEMBL23968103 0.85 MELK (0.46) MAPKAPK2MELKKMT2ATGFBR1MEN1
SCHEMBL23968014 0.84 MELK (0.45) MAPKAPK2MELK
SCHEMBL23968072 0.84 MELK (0.45) MAPKAPK2MELK
SCHEMBL23968093 0.83 MAP4K4 (0.54) MELKRAB9ANPC1MAPTALDH1A1
SCHEMBL23968001 0.83 MELK (0.51) MELKMAPTALDH1A1GRM4
SCHEMBL23968101 0.81 DRD2 (0.43) MAPKAPK2MELKRAB9ANPC1HTR3E
SCHEMBL902160 0.80 HTR3E (0.61) RAB9ANPC1HTR3EHTR3BADRB1
SCHEMBL23968090 0.80 MELK (0.49) MAPKAPK2MELKMAPTALDH1A1
SCHEMBL23968098 0.80 MELK (0.48) MELKRAB9ANPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2021-11-03 EP disclosed