SCHEMBL23968101

SCHEMBL23968101

COc1ccccc1-n1cc(-c2ccc(N3CCSCC3)cc2)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.43
DRD3 P35462 7/20 0.43
DRD4 P21917 5/20 0.43
HTR1A P08908 4/20 0.43
MELK Q14680 2/20 0.43
DYRK1B Q9Y463 1/20 0.41
MTOR P42345 2/20 0.41
MAPT P10636 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NMT1 P30419 1/20 0.39
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23968161 0.85 S1PR1 (0.41) DRD2DRD3DRD4HTR1AMELK
SCHEMBL23968179 0.82 GRM4 (0.44) DRD2DRD3DRD4MELKDYRK1B
SCHEMBL23968008 0.82 MELK (0.41) DRD2DRD3DRD4MELKMTOR
SCHEMBL23968199 0.81 MAPKAPK2 (0.57) MELKMAPTSMN1; SMN2KDM4ENPC1
SCHEMBL7805608 0.79 AVPR2 (0.49) DRD2DRD3DRD4HTR1ADYRK1B
SCHEMBL23968113 0.79 MELK (0.39) DRD2DRD3DRD4MELK
SCHEMBL23968136 0.79 MKNK1 (0.47) MELKMAPTNMT1KDM4ENPC1
SCHEMBL23968184 0.79 MELK (0.39) MELK
SCHEMBL23968103 0.79 MELK (0.46) MELKMTORMEN1KMT2AMAPKAPK2
SCHEMBL23968001 0.76 MELK (0.51) DRD2DRD3DRD4MELKMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2021-11-03 EP disclosed