SCHEMBL23968115

SCHEMBL23968115

Fc1cnc(-n2cc(-c3ccc(N4CCSCC4)cc3)cn2)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.42
MELK Q14680 2/20 0.38
CNR2 P34972 1/20 0.34
EGLN1 Q9GZT9 1/20 0.34
KCNH2 Q12809 1/20 0.34
MAPT P10636 2/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAP4K4 O95819 1/20 0.33
JAK2 O60674 1/20 0.32
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32
AR P10275 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CTSC P53634 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23968105 0.89 MELK (0.39) POLBMELKEGLN1MAPTDRD2
SCHEMBL23968168 0.80 MELK (0.46) MELKEGLN1MAPTMAP4K4DRD2
SCHEMBL23968001 0.80 MELK (0.51) MELKMAPTHTTMAP4K4DRD2
SCHEMBL23967998 0.79 MELK (0.41) MELKCNR2EGLN1MAPTDRD2
SCHEMBL23968153 0.77 MELK (0.42) MELKEGLN1MAPT
SCHEMBL23968093 0.77 MAP4K4 (0.54) POLBMELKKCNH2MAPTSMN1; SMN2
SCHEMBL23968099 0.77 GRM4 (0.46) MELKEGLN1DRD2DRD4DRD3
SCHEMBL23968162 0.76 MELK (0.40) MELKMAPTHTTSMN1; SMN2DRD2
SCHEMBL23968157 0.76 MELK (0.40) MELKEGLN1KCNH2MAPTDRD2
SCHEMBL23968008 0.75 MELK (0.41) MELKCNR2EGLN1MAPTMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2021-11-03 EP disclosed