SCHEMBL23970519

SCHEMBL23970519

CC(C)COC(=O)c1cnn(C)c1Br

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
TSHR P16473 1/20 0.50
JMJD6 Q6NYC1 1/20 0.38
NPC1 O15118 4/20 0.37
RAB9A P51151 4/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 2/20 0.37
HTT P42858 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MEN1 O00255 1/20 0.36
TP53 P04637 1/20 0.36
NPY1R P25929 1/20 0.36
NPY2R P49146 1/20 0.36
KMT2A Q03164 1/20 0.36
ATM Q13315 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PLA2G1B P04054 1/20 0.35
ATG4B Q9Y4P1 1/20 0.35
ADRA1D P25100 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2315523 0.83 RAB9A (0.48) ALDH1A1TSHRNPC1RAB9ASMN1; SMN2
SCHEMBL26654708 0.77 CYP1A2 (0.49) ALDH1A1TSHRNPC1RAB9ASMN1; SMN2
SCHEMBL23970512 0.74 ALDH1A1 (0.42) ALDH1A1TSHRJMJD6NPC1RAB9A
SCHEMBL30696931 0.73 RAB9A (0.45) ALDH1A1TSHRNPC1RAB9ASMN1; SMN2
SCHEMBL11971062 0.72 SMN1; SMN2 (0.40) ALDH1A1NPC1RAB9ASMN1; SMN2HTT
SCHEMBL4628560 0.72 TSHR (0.61) ALDH1A1TSHRJMJD6NPC1RAB9A
SCHEMBL23970517 0.72 ALDH1A1 (0.40) ALDH1A1TSHRJMJD6NPC1RAB9A
SCHEMBL826742 0.71 SMN1; SMN2 (0.41) ALDH1A1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL827863 0.70 TSHR (0.70) ALDH1A1TSHRJMJD6NPC1RAB9A
SCHEMBL23693030 0.70 ALDH1A1 (0.42) ALDH1A1TSHRJMJD6NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222353-A1 MACROCYCLIC INHIBITORS OF PEPTIDYLARGININE DEIMINASES GILEAD SCIENCES, INC. (US) 2021-11-04 WO disclosed