SCHEMBL23972253

SCHEMBL23972253

CC1=CCN(C(=O)C2CCC(C(F)(F)F)CC2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.39
HSD11B1 P28845 1/20 0.37
JAK1 P23458 3/20 0.36
ALDH1A1 P00352 2/20 0.36
NAMPT P43490 1/20 0.36
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
GAA P10253 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
KEAP1 Q14145 1/20 0.36
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
MAPT P10636 3/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
SPR P35270 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
TP53 P04637 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17342884 0.88 KEAP1 (0.43) JAK1ALDH1A1NAMPTKDM4EUSP2
SCHEMBL26027615 0.83 NR1H2 (0.37) GRM5HSD11B1JAK1ALDH1A1KDM4E
SCHEMBL17888264 0.82 KEAP1 (0.51) HSD11B1ALDH1A1NAMPTTSHRKEAP1
SCHEMBL19226370 0.82 KEAP1 (0.48) HSD11B1ALDH1A1NAMPTTSHRKEAP1
SCHEMBL17888277 0.81 KEAP1 (0.54) HSD11B1ALDH1A1NAMPTTSHRKEAP1
SCHEMBL7920857 0.80 NAMPT (0.47) GRM5ALDH1A1NAMPTKDM4EKEAP1
SCHEMBL12286462 0.79 MAPT (0.37) JAK1ALDH1A1NAMPTKDM4EUSP2
SCHEMBL17888258 0.78 NAMPT (0.51) GRM5ALDH1A1NAMPTKDM4ETSHR
SCHEMBL12286226 0.78 CHRNB2 (0.46) JAK1ALDH1A1NAMPTKDM4EUSP2
SCHEMBL17888278 0.78 JAK1 (0.38) GRM5JAK1ALDH1A1NAMPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021221169-A1 PYRIMIDIN-4(3H)-ONE DERIVATIVES AS TRPV4 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2021-11-04 WO disclosed