SCHEMBL2397288

SCHEMBL2397288

Cc1nc(Nc2cc[nH]n2)sc1-c1ccc(Cl)c(S(=O)(=O)N(CCO)CCO)c1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PI4KB Q9UBF8 14/20 0.49
PIK3CD O00329 7/20 0.49
PIK3CG P48736 7/20 0.49
PIK3C3 Q8NEB9 3/20 0.49
PIK3CA P42336 2/20 0.49
PIK3CB P42338 2/20 0.49
PIK3C2A O00443 1/20 0.49
PIK3C2B O00750 1/20 0.49
PI4KA P42356 1/20 0.49
PRKDC P78527 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2396778 0.85 PIK3CD (0.68) PI4KBPIK3CDPIK3CGPIK3C3PIK3CA
SCHEMBL2398836 0.81 PIK3CD (0.54) PI4KBPIK3CDPIK3CGPIK3C3PIK3CA
SCHEMBL48507 0.75 PIK3CD (0.57) PI4KBPIK3CDPIK3CGPIK3C3PIK3CA
SCHEMBL2396380 0.73 PIK3CD (0.62) PI4KBPIK3CDPIK3CGPIK3C3PIK3CA
SCHEMBL2397182 0.72 PIK3CD (0.49) PI4KBPIK3CDPIK3CGPIK3C3PIK3CA
Bromide SCHEMBL2398769 0.72 PIK3CD (0.61) PI4KBPIK3CDPIK3CGPIK3C3PIK3CA
SCHEMBL49344 0.72 PIK3CD (0.59) PI4KBPIK3CDPIK3CGPIK3C3PIK3CA
SCHEMBL2398248 0.71 PIK3CD (0.40) PI4KBPIK3CDPIK3CGPIK3CAPIK3CB
SCHEMBL1886940 0.71 NPC1 (0.39) PI4KBPIK3CDPIK3CGPIK3C3PIK3CA
SCHEMBL2397832 0.71 MEN1 (0.61) PIK3CDPIK3CGPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8017608-B2 5-Phenylthiazole derivatives and their use as p13 kinase inhibitors NOVARTIS AG (CH) 2011-09-13 US disclosed
EP-1608647-B1 5-PHENYLTHIAZOLE DERIVATIVES AND THEIR USE AS P13 KINASE INHIBITORS NOVARTIS AG (CH) 2008-01-09 EP disclosed
US-20060148822-A1 5-Phenylthiazole derivatives and their use as p13 kinase inhibitors NOVARTIS AG (CH) 2006-07-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060148822-A1 5-Phenylthiazole derivatives and their use as p13 kinase inhibitors MAP3K13, AKT3, MAP3K3 PI4KB 56/4885PIK3CD 42/4885PIK3CG 49/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.