SCHEMBL2397562

SCHEMBL2397562

COc1ccc(NC2CCN(C(=O)N(C)c3ccc(CN4CCN(C(=O)O)[C@@](C)(C(C)(C)C)C4)cc3)CC2)cc1F

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MLNR O43193 11/20 0.39
CYP3A4 P08684 4/20 0.37
FAAH O00519 1/20 0.36
MCHR1 Q99705 2/20 0.35
UBE2M P61081 1/20 0.35
DCUN1D1 Q96GG9 1/20 0.35
KCNH2 Q12809 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
GALR3 O60755 1/20 0.35
RAB9A P51151 1/20 0.35
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL377748 0.87 MLNR (0.49) MLNRCYP3A4FAAHKCNH2
SCHEMBL377854 0.84 MLNR (0.47) MLNRCYP3A4FAAHRORC
SCHEMBL377818 0.82 MLNR (0.46) MLNRCYP3A4KCNH2
SCHEMBL2397561 0.79 MLNR (0.44) MLNRCYP3A4KCNH2RAB9A
SCHEMBL377498 0.79 MLNR (0.64) MLNRCYP3A4KCNH2
SCHEMBL2393780 0.78 FAAH (0.40) MLNRCYP3A4FAAHRORC
SCHEMBL377770 0.78 CHRM4 (0.42) MLNRFAAHMCHR1SIGMAR1
SCHEMBL2396382 0.78 MLNR (0.43) MLNRCYP3A4FAAHRORC
SCHEMBL376913 0.78 MLNR (0.40) MLNRCYP3A4FAAHKCNH2
SCHEMBL377719 0.78 MLNR (0.40) MLNRCYP3A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012981-B2 Benzylpiperazine derivatives as motilin receptor agonists GLAXO GROUP LIMITED (GB) 2011-09-06 US disclosed