SCHEMBL2393780

SCHEMBL2393780

CN(C(=O)N1CCC(Nc2ccccc2C(N)=O)CC1)c1ccc(CN2CCN(C(=O)O)[C@@](C)(C(C)(C)C)C2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.40
MLNR O43193 3/20 0.36
CYP3A4 P08684 2/20 0.36
PARP1 P09874 1/20 0.35
OPRD1 P41143 2/20 0.35
OPRM1 P35372 1/20 0.35
DRD4 P21917 1/20 0.35
RORC P51449 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
JAK3 P52333 1/20 0.34
HSP90AA1 P07900 1/20 0.34
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
OPRK1 P41145 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2396382 0.87 MLNR (0.43) FAAHMLNRCYP3A4DRD4RORC
SCHEMBL377748 0.82 MLNR (0.49) FAAHMLNRCYP3A4KDM4EALDH1A1
SCHEMBL377854 0.82 MLNR (0.47) FAAHMLNRCYP3A4RORC
SCHEMBL377935 0.81 FAAH (0.42) FAAHMLNRCYP3A4PARP1DRD4
SCHEMBL2397562 0.78 MLNR (0.39) FAAHMLNRCYP3A4RORC
SCHEMBL377770 0.77 CHRM4 (0.42) FAAHMLNR
SCHEMBL377479 0.77 MLNR (0.49) MLNRCYP3A4
SCHEMBL2393775 0.77 BRD4 (0.39) FAAHMLNRCYP3A4PARP1ALDH1A1
SCHEMBL377588 0.76 CHRM4 (0.45) FAAHMLNRDRD4MEN1KMT2A
SCHEMBL2397558 0.76 MLNR (0.46) FAAHMLNRMEN1KMT2AOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012981-B2 Benzylpiperazine derivatives as motilin receptor agonists GLAXO GROUP LIMITED (GB) 2011-09-06 US disclosed