SCHEMBL23976125

SCHEMBL23976125

CN(C)CCOc1ccnc(-c2nc3c(c(N(C)CC(N)=O)n2)CCC3)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.36
HDAC1 Q13547 5/20 0.36
HDAC8 Q9BY41 4/20 0.36
HDAC6 Q9UBN7 4/20 0.36
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 2/20 0.35
PDE10A Q9Y233 1/20 0.35
NOS3 P29474 2/20 0.35
NOS1 P29475 2/20 0.35
NOS2 P35228 2/20 0.35
SPR P35270 1/20 0.34
DYRK3 O43781 1/20 0.33
MAP4K4 O95819 1/20 0.33
PIM1 P11309 1/20 0.33
RPS6KB1 P23443 1/20 0.33
CSNK2A1 P68400 1/20 0.33
PKN2 Q16513 1/20 0.33
PIM3 Q86V86 1/20 0.33
BRSK1 Q8TDC3 1/20 0.33
AURKB Q96GD4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23975592 0.92 SYK (0.38) HDAC1HDAC8HDAC6PDE10ASPR
SCHEMBL23976123 0.92 KDM4E (0.38) PARP1HDAC1HDAC8HDAC6KDM4E
SCHEMBL30484199 0.90 TUBB3 (0.38) HDAC1HDAC8HDAC6KDM4EALDH1A1
SCHEMBL23975862 0.90 TUBB3 (0.38) HDAC1HDAC8HDAC6KDM4EALDH1A1
Formic Acid SCHEMBL30225275 0.89 KDM4E (0.36) PARP1HDAC1HDAC8HDAC6KDM4E
SCHEMBL23987002 0.89 KDM4E (0.36) PARP1HDAC1HDAC8HDAC6KDM4E
SCHEMBL23976372 0.88 HDAC1 (0.38) PARP1HDAC1HDAC8HDAC6KDM4E
SCHEMBL23976947 0.88 PDE10A (0.38) PARP1HDAC1HDAC8HDAC6KDM4E
SCHEMBL23976139 0.87 HDAC1 (0.37) PARP1HDAC1HDAC8HDAC6KDM4E
SCHEMBL23976413 0.86 HDAC1 (0.33) HDAC1HDAC8HDAC6PDE10ASPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222483-A1 METHODS OF USE FOR PYRIMIDINES AS FERROPORTIN INHIBITORS GLOBAL BLOOD THERAPEUTICS, INC. (US) 2021-11-04 WO disclosed
WO-2021222363-A1 CYCLOALKYL PYRIMIDINES AS FERROPORTIN INHIBITORS GLOBAL BLOOD THERAPEUTICS, INC. (US) 2021-11-04 WO disclosed